Cargando…

QSAR Analysis of Benzophenone Derivatives as Antimalarial Agents

A set of benzophenone derivatives was evaluated for the antimalarial activity against Plasmodium berghei in mice and the mean survival time of mice for all the compounds was determined. The QSAR analysis was carried out for the fourteen benzophenone derivatives using different physicochemical descri...

Descripción completa

Detalles Bibliográficos
Autores principales:	Mahajan, Supriya, Kamath, Vijayalaxmi, Nayak, Sonali, Vaidya, Shalaka
Formato:	Online Artículo Texto
Lenguaje:	English
Publicado:	Medknow Publications & Media Pvt Ltd 2012
Materias:	Research Paper
Acceso en línea:	https://www.ncbi.nlm.nih.gov/pmc/articles/PMC3507344/ https://www.ncbi.nlm.nih.gov/pubmed/23204621 http://dx.doi.org/10.4103/0250-474X.102542

Ejemplares similares

QSAR Study of N-Myristoyltransferase Inhibitors of Antimalarial Agents
por: Santos-Garcia, Letícia, et al.
Publicado: (2018)

3D-QSAR, docking and ADMET properties of aurone analogues as antimalarial agents
por: Hadni, Hanine, et al.
Publicado: (2020)

Classical QSAR and Docking Simulation of 4-Pyridone Derivatives for Their Antimalarial Activity
por: Flores-Sumoza, Máryury, et al.
Publicado: (2018)

Derivative spectrophotometric analysis of benzophenone (as an impurity) in phenytoin
por: Walash, Mohamed Ibrahim, et al.
Publicado: (2011)

Novel series of 1,2,4-trioxane derivatives as antimalarial agents
por: Rudrapal, Mithun, et al.
Publicado: (2017)

Theoretical design of novel antimalarial agents against P. falciparum strain, Dd(2) through the QSAR modeling of synthesized 2′-substituted triclosan derivatives
por: Ibrahim, Zakari Ya'u, et al.
Publicado: (2020)

A SAR and QSAR Study of New Artemisinin Compounds with Antimalarial Activity
por: Santos, Cleydson Breno R., et al.
Publicado: (2013)

An alternative to hydrogenation processes. Electrocatalytic hydrogenation of benzophenone
por: Mozo Mulero, Cristina, et al.
Publicado: (2018)

Benzophenone-3 promotion of mammary tumorigenesis is diet-dependent
por: Kariagina, Anastasia, et al.
Publicado: (2020)

New Potential Antimalarial Agents: Design, Synthesis and Biological Evaluation of Some Novel Quinoline Derivatives as Antimalarial Agents
por: Radini, Ibrahim Ali M., et al.
Publicado: (2016)

Three New Benzophenone Derivatives from Selaginella tamariscina
por: Long, Jiayin, et al.
Publicado: (2023)

Evaluation by the Ames Assay of the Mutagenicity of UV Filters Using Benzophenone and Benzophenone-1
por: Wang, Wen-Qian, et al.
Publicado: (2018)

QSAR-Based Virtual Screening of Natural Products Database for Identification of Potent Antimalarial Hits
por: Ferreira, Letícia Tiburcio, et al.
Publicado: (2021)

Heavy atom effects in the Paternò–Büchi reaction of pyrimidine derivatives with 4,4’-disubstituted benzophenones
por: Kong, Feng-Feng, et al.
Publicado: (2011)

4,4′-Dimethoxybenzophenone: a triclinic polymorph
por: Fun, Hoong-Kun, et al.
Publicado: (2008)

Ferroquine and its derivatives: New generation of antimalarial agents
por: Wani, Waseem A., et al.
Publicado: (2015)

Advantages and limitations of classic and 3D QSAR approaches in nano-QSAR studies based on biological activity of fullerene derivatives
por: Jagiello, Karolina, et al.
Publicado: (2016)

In-silico combinatorial design and pharmacophore modeling of potent antimalarial 4-anilinoquinolines utilizing QSAR and computed descriptors
por: Parihar, Neha, et al.
Publicado: (2015)

Mutagenicity evaluation to UV filters of benzophenone-6, benzophenone-8, and 4-methylbenzylidene camphor by Ames test
por: Zhang, Jing, et al.
Publicado: (2021)

Structure–Activity Relationship Studies of Pyrrolone Antimalarial Agents
por: Murugesan, Dinakaran, et al.
Publicado: (2013)

Synthesis and Evaluation of Benzophenone-N-ethyl Morpholine Ethers as Anti-inflammatory Agents
por: Khanum, Shaukath A., et al.
Publicado: (2010)

Prenylated Benzophenones from Vismia Guianensis Reduced Nematode Growth and Chemotaxis
por: Gerald, Carresse, et al.
Publicado: (2023)

Safety of benzophenone to be used as flavouring
por: Silano, Vittorio, et al.
Publicado: (2017)

New pyrazolylpyrazoline derivatives as dual acting antimalarial-antileishamanial agents: synthesis, biological evaluation and molecular modelling simulations
por: Bekhit, Adnan A., et al.
Publicado: (2022)

Application of QSAR Method in the Design of Enhanced Antimalarial Derivatives of Azetidine-2-carbonitriles, their Molecular Docking, Drug-likeness, and SwissADME Properties
por: Ibrahim, Zakari Ya’u, et al.
Publicado: (2021)

Benzophenone Derivatives from an Algal-Endophytic Isolate of Penicillium chrysogenum and Their Cytotoxicity
por: Zhao, Dong-Lin, et al.
Publicado: (2018)

Light-Assisted Synthesis of Silver and Gold Nanoparticles by New Benzophenone Derivatives
por: Alnafisah, Abrar S., et al.
Publicado: (2023)

3D-QSAR CoMFA study of some Heteroarylpyrroles as Possible Anticandida Agents
por: Sharma, P. C., et al.
Publicado: (2008)

Fate of Benzophenone, Benzophenone-3 and Caffeine in Lab-Scale Direct River Water Treatment by Hybrid Processes
por: Bogunović, Minja, et al.
Publicado: (2021)

Toxicokinetics, Percutaneous Absorption and Tissue Distribution of Benzophenone-3, an UV Filtering Agent, in Rats
por: Jung, Woohyung, et al.
Publicado: (2022)

Hammett correlation in competition experiments in dissociation of ionised substituted benzophenones and dibenzylideneacetones
por: Fenwick, Nathan W, et al.
Publicado: (2023)

Discovery of novel benzophenone integrated derivatives as anti-Alzheimer’s agents targeting presenilin-1 and presenilin-2 inhibition: A computational approach
por: Martiz, Reshma Mary, et al.
Publicado: (2022)

New benzophenone and quercetin galloyl glycosides from Psidium guajava L.
por: Matsuzaki, Keiichi, et al.
Publicado: (2010)

4-Chloro-2′,4′,6′-triethylbenzophenone: a redetermination
por: Takahashi, Hiroki
Publicado: (2011)

QSAR Study on Thiazolidine-2,4-dione Derivatives for Antihyperglycemic Activity
por: Prashantha Kumar, B. R., et al.
Publicado: (2008)

Benzophenones in the Environment: Occurrence, Fate and Sample Preparation in the Analysis
por: Gavrila, Andromachi A., et al.
Publicado: (2023)

Molecular docking and QSAR studies for modeling the antimalarial activity of hybrids 4-anilinoquinoline-triazines derivatives with the wild-type and mutant receptor pf-DHFR
por: Hadni, Hanine, et al.
Publicado: (2019)

Design, synthesis, biological evaluation and QSAR analysis of novel N-substituted benzimidazole derived carboxamides
por: Beč, Anja, et al.
Publicado: (2022)

Antimalarial properties and molecular docking analysis of compounds from Dioscorea bulbifera L. as new antimalarial agent candidates
por: Chaniad, Prapaporn, et al.
Publicado: (2021)

New 1-Aryl-3-Substituted Propanol Derivatives as Antimalarial Agents
por: Pérez-Silanes, Silvia, et al.
Publicado: (2009)

Cannot write session to /tmp/vufind_sessions/sess_ldh6mncdmp4uivg5f7qdm96ou7