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Synthesis of 5-oxyquinoline derivatives for reversal of multidrug resistance

The inhibition of ABC (ATP binding cassette) transporters is considered a powerful tool to reverse multidrug resistance. Zosuquidar featuring a difluorocyclopropyl-annulated dibenzosuberyl moiety has been found to be an inhibitor of the P-glycoprotein, one of the best-studied multidrug efflux pumps....

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Detalles Bibliográficos
Autores principales:	Dittrich, Torsten, Hanekop, Nils, Infed, Nacera, Schmitt, Lutz, Braun, Manfred
Formato:	Online Artículo Texto
Lenguaje:	English
Publicado:	Beilstein-Institut 2012
Materias:	Full Research Paper
Acceso en línea:	https://www.ncbi.nlm.nih.gov/pmc/articles/PMC3511002/ https://www.ncbi.nlm.nih.gov/pubmed/23209502 http://dx.doi.org/10.3762/bjoc.8.193

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