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An easy direct arylation of 5-pyrazolones

A mild, efficient and catalytic ligand-free method for the direct arylation of 5-pyrazolones by Pd-catalyzed C–H bond activation is reported. The process smoothly proceeds and yields are moderate to excellent.

Detalles Bibliográficos
Autores principales:	Gong, Hao, Yang, Yiwen, Wang, Zechao, Kuang, Chunxiang
Formato:	Online Artículo Texto
Lenguaje:	English
Publicado:	Beilstein-Institut 2013
Materias:	Full Research Paper
Acceso en línea:	https://www.ncbi.nlm.nih.gov/pmc/articles/PMC3817516/ https://www.ncbi.nlm.nih.gov/pubmed/24204415 http://dx.doi.org/10.3762/bjoc.9.240

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