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Structure-Activity Relationships of Constrained Phenylethylamine Ligands for the Serotonin 5-HT(2) Receptors

Serotonergic ligands have proven effective drugs in the treatment of migraine, pain, obesity, and a wide range of psychiatric and neurological disorders. There is a clinical need for more highly 5-HT(2) receptor subtype-selective ligands and the most attention has been given to the phenethylamine cl...

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Detalles Bibliográficos
Autores principales:	Isberg, Vignir, Paine, James, Leth-Petersen, Sebastian, Kristensen, Jesper L., Gloriam, David E.
Formato:	Online Artículo Texto
Lenguaje:	English
Publicado:	Public Library of Science 2013
Materias:	Research Article
Acceso en línea:	https://www.ncbi.nlm.nih.gov/pmc/articles/PMC3820707/ https://www.ncbi.nlm.nih.gov/pubmed/24244317 http://dx.doi.org/10.1371/journal.pone.0078515

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