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Synthesis and Evaluation of [(67)Ga]-AMD3100: A Novel Imaging Agent for Targeting the Chemokine Receptor CXCR4
In order to develop a possible C-X-C chemokine receptor type 4 (CXCR4) imaging agent for oncological scintigraphy, [(67)Ga]-labeled 1,1′-[1,4-Phenylene-bis(methylene)]bis(1,4,8,11-tetraazacyclotetradecane) ([(67)Ga]-AMD3100) was prepared by using [(67)Ga]GaCl(3) and AMD-3100 for 2 h at 50 °C (radioc...
Autores principales: | Aghanejad, Ayuob, Jalilian, Amir R., Fazaeli, Yousef, Alirezapoor, Behrouz, Pouladi, Mehraban, Beiki, Davoud, Maus, Stephan, Khalaj, Ali |
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Formato: | Online Artículo Texto |
Lenguaje: | English |
Publicado: |
Österreichische Apotheker-Verlagsgesellschaft
2014
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Materias: | |
Acceso en línea: | https://www.ncbi.nlm.nih.gov/pmc/articles/PMC3951231/ https://www.ncbi.nlm.nih.gov/pubmed/24634840 http://dx.doi.org/10.3797/scipharm.1305-18 |
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