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Arylation and Heteroarylation of Thienylsulfonamides with Organotrifluoroborates

[Image: see text] A mild, practical protocol has been developed for the Suzuki cross-coupling of unprotected thienylsulfonamides from air- and bench-stable organotrifluoroborates in the absence of a protecting group on the sulfonamide nitrogen. The developed synthetic method can be applied to the pr...

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Detalles Bibliográficos
Autores principales:	Noreen, Mnaza, Rasool, Nasir, El Khatib, Mirna, Molander, Gary A.
Formato:	Online Artículo Texto
Lenguaje:	English
Publicado:	American Chemical Society 2014
Acceso en línea:	https://www.ncbi.nlm.nih.gov/pmc/articles/PMC4120984/ https://www.ncbi.nlm.nih.gov/pubmed/25019222 http://dx.doi.org/10.1021/jo501323z

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