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Regioselective Synthesis of Benzimidazolones via Cascade C–N Coupling of Monosubstituted Ureas

[Image: see text] A direct method for the regioselective construction of benzimidazolones is reported wherein a single palladium catalyst is employed to couple monosubstituted urea substrates with differentially substituted 1,2-dihaloaromatic systems. In this method, the catalyst is able to promote...

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Detalles Bibliográficos
Autores principales:	Ernst, Johannes B., Tay, Nicholas E. S., Jui, Nathan T., Buchwald, Stephen L.
Formato:	Online Artículo Texto
Lenguaje:	English
Publicado:	American Chemical Society 2014
Acceso en línea:	https://www.ncbi.nlm.nih.gov/pmc/articles/PMC4216194/ https://www.ncbi.nlm.nih.gov/pubmed/24971635 http://dx.doi.org/10.1021/ol501531q

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