Cargando…

Antimicrobial screening and one-pot synthesis of 4-(substituted-anilinomethyl)-3-(2-naphthyl)-1-phenyl-1H-pyrazole derivatives

AIM: Synthesis of series of 4-(substituted-anilinomethyl-3-(2-naphthyl)-1-phenyl-1H-pyrazole derivatives (4a–4k) and their in vitro antifungal and antibacterial screening. MATERIALS AND METHODS: A series of compounds (4a–4k) was synthesized through direct reductive amination of 3-(naphthalen-2-yl)-1...

Descripción completa

Detalles Bibliográficos
Autores principales:	Goel, Neelima, Drabu, Sushma, Afzal, Obaid, Bawa, Sandhya
Formato:	Online Artículo Texto
Lenguaje:	English
Publicado:	Medknow Publications & Media Pvt Ltd 2014
Materias:	Original Article
Acceso en línea:	https://www.ncbi.nlm.nih.gov/pmc/articles/PMC4231385/ https://www.ncbi.nlm.nih.gov/pubmed/25400408 http://dx.doi.org/10.4103/0975-7406.142956

Ejemplares similares

Development of 4-[4-(Anilinomethyl)-3-phenyl-pyrazol-1-yl] Benzoic Acid Derivatives as Potent Anti-Staphylococci and Anti-Enterococci Agents
por: Raj KC, Hansa, et al.
Publicado: (2022)

Synthesis and biological evaluation of di- and tri-substituted imidazoles as safer anti-inflammatory-antifungal agents
por: Husain, Asif, et al.
Publicado: (2013)

3-Anilinomethyl-5-chloro-1,3-benzoxazol-2(3H)-one
por: Aydın, Abdullah, et al.
Publicado: (2012)

Structural modifications of quinoline-based antimalarial agents: Recent developments
por: Bawa, Sandhya, et al.
Publicado: (2010)

4-[(Z)-(2-Furyl)(2-naphthylamino)methylene)]-3-methyl-1-phenyl-1H-pyrazol-5(4H)-one
por: Li, Jing, et al.
Publicado: (2009)

1-(2-Naphthyl)-3-phenylprop-2-en-1-one
por: Tang, Si-Ping, et al.
Publicado: (2009)

4-[(1-Hydroxy-2-naphthyl)methyleneamino]-1,5-dimethyl-2-phenyl-1H-pyrazol-3(2H)-one
por: Liang, Qiang, et al.
Publicado: (2010)

4-[(Z)-(2-Furyl)(2-naphthylamino)methylene)]-3-methyl-1-phenyl-1H-pyrazol-5(4H)-one. Corrigendum
por: Li, Jing, et al.
Publicado: (2010)

6-(2-Hydroxyanilinomethylene)-4-nitrocyclohexa-2,4-dien-1-one
por: Böhme, Uwe, et al.
Publicado: (2007)

3-(1-Naphthyl)-N-phenyloxirane-2-carboxamide
por: Chen, Lian-Mei, et al.
Publicado: (2009)

Design, synthesis, molecular modelling and biological evaluation of novel 3-(2-naphthyl)-1-phenyl-1H-pyrazole derivatives as potent antioxidants and 15-Lipoxygenase inhibitors
por: Ali, Sahar A., et al.
Publicado: (2020)

Catalyst-Free One-Pot Synthesis of Densely Substituted Pyrazole-Pyrazines as Anti-Colorectal Cancer Agents
por: Xu, Jia, et al.
Publicado: (2020)

Synthesis, characterization, and biological evaluation of new copper complexes of naphthyl pyrazole ligands
por: HINIS, Melek, et al.
Publicado: (2021)

2-[2-(Hydroxymethyl)phenyl]-1-(1-naphthyl)ethanol
por: Khan, F. Nawaz, et al.
Publicado: (2010)

1-Phenyl-1H-pyrazole-4-carbaldehyde
por: Asiri, Abdullah M., et al.
Publicado: (2012)

Bis[5-(2-naphthyl)-1H-pyrazole-κN (2)]silver(I) nitrate
por: Wang, Zhao-Yang, et al.
Publicado: (2009)

Chiral Chalcogenyl‐Substituted Naphthyl‐ and Acenaphthyl‐Silanes and Their Cations
por: Künzler, Sandra, et al.
Publicado: (2020)

A One-Pot Divergent Sequence to Pyrazole and Quinoline Derivatives
por: Gambacorta, Guido, et al.
Publicado: (2020)

5-(4-Bromoanilinomethylene)-2,2-dimethyl-1,3-dioxane-4,6-dione
por: Shi, Jian-You, et al.
Publicado: (2009)

5-(4-Chloroanilinomethylene)-2,2-dimethyl-1,3-dioxane-4,6-dione
por: Yang, Jin-Cheng, et al.
Publicado: (2009)

3-Acetyl-1-(3-methylphenyl)-5-phenyl-1H-pyrazole-4-carbonitrile
por: Abdel-Aziz, Hatem A., et al.
Publicado: (2012)

[2-(2-Methoxy-1-naphthoyl)phenyl](1-naphthyl)methanone
por: Jagadeesan, G., et al.
Publicado: (2011)

5-Acetyl-3-(5-phenyl-1H-pyrazol-3-yl)-1,3,4-thiadiazol-2(3H)-one monohydrate
por: Asiri, Abdullah M., et al.
Publicado: (2013)

N-[(2-Hydroxy-1-naphthyl)(3-nitrophenyl)methyl]acetamide
por: NizamMohideen, M., et al.
Publicado: (2009)

5-(Adamantan-1-yl)-3-anilinomethyl-2,3-dihydro-1,3,4-oxadiazole-2-thione
por: Al-Tamimi, Abdul-Malek S., et al.
Publicado: (2013)

3-Methyl-5-phenyl-1-(3-phenylisoquinolin-1-yl)-1H-pyrazole
por: Khan, F. Nawaz, et al.
Publicado: (2010)

Synthesis, biological evaluation and in silico molecular docking of novel 1-hydroxy-naphthyl substituted heterocycles
por: El-Desoky, El-Sayed I., et al.
Publicado: (2018)

(8-Bromo-2,7-dimethoxy-1-naphthyl)(4-chlorophenyl)methanone
por: Mitsui, Ryosuke, et al.
Publicado: (2010)

Synthesis and Antifungal Activity of N-(Substituted pyridinyl)-1-methyl(phenyl)-3-(trifluoromethyl)-1H-pyrazole-4-carboxamide Derivatives
por: Wu, Zhibing, et al.
Publicado: (2012)

1-(2,4-Dinitrophenyl)-3-(4-methylphenyl)-4-phenylsulfanyl-1H-pyrazole
por: Ramesh, P., et al.
Publicado: (2008)

5-Chloro-1-phenyl-1H-pyrazol-4-amine
por: Korzański, Artur, et al.
Publicado: (2011)

Enaminones as Building Blocks for the Synthesis of Substituted Pyrazoles with Antitumor and Antimicrobial Activities
por: Riyadh, Sayed M.
Publicado: (2011)

Antimicrobial screening to molecular docking of newly synthesized ferrocenyl-substituted pyrazole
por: Sharma, Shashi, et al.
Publicado: (2022)

4-[(5-Hydroxy-3-methyl-1-phenyl-1H-pyrazol-4-yl)phenylmethyl]-5-methyl-2-phenyl-1H-pyrazol-3(2H)-one ethanol hemisolvate
por: Fun, Hoong-Kun, et al.
Publicado: (2008)

4-Methyl-5-phenyl-1H-pyrazol-3(2H)-one
por: Loh, Wan-Sin, et al.
Publicado: (2010)

5-Ethyl-4-phenyl-1H-pyrazol-3(2H)-one
por: Loh, Wan-Sin, et al.
Publicado: (2011)

(E)-3-Phenyl-3-(3-phenyl-1H-1-pyrazolyl)-2-propenal
por: Susindran, V., et al.
Publicado: (2010)

(E)-5-Phenyl-N′-(1-phenylethylidene)-1H-pyrazole-3-carbohydrazide
por: Qin, Yongqi, et al.
Publicado: (2007)

3-Methyl-1-phenyl-4-[(phenyl)(2-phenylhydrazin-1-yl)methylidene]-1H-pyrazol-5(4H)-one
por: Idemudia, Omoruyi G., et al.
Publicado: (2012)

4-{[(E)-(3,5-Dimethyl-1-phenyl-1H-pyrazol-4-yl)methylidene]amino}-1,5-dimethyl-2-phenyl-1H-pyrazol-3(2H)-one
por: Fun, Hoong-Kun, et al.
Publicado: (2010)

Cannot write session to /tmp/vufind_sessions/sess_u6oicrgshl4d6jeipu9rmqm71l