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3D QSAR Studies, Pharmacophore Modeling and Virtual Screening on a Series of Steroidal Aromatase Inhibitors

Aromatase inhibitors are the most important targets in treatment of estrogen-dependent cancers. In order to search for potent steroidal aromatase inhibitors (SAIs) with lower side effects and overcome cellular resistance, comparative molecular field analysis (CoMFA) and comparative molecular similar...

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Detalles Bibliográficos
Autores principales:	Xie, Huiding, Qiu, Kaixiong, Xie, Xiaoguang
Formato:	Online Artículo Texto
Lenguaje:	English
Publicado:	MDPI 2014
Materias:	Article
Acceso en línea:	https://www.ncbi.nlm.nih.gov/pmc/articles/PMC4264204/ https://www.ncbi.nlm.nih.gov/pubmed/25405729 http://dx.doi.org/10.3390/ijms151120927

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