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Synthesis and molecular docking of novel non-competitive antagonists of GluK2 receptor
Here we present the synthesis, pharmacological activity, and molecular docking of novel non-competitive antagonists of GluK2 receptor. The compounds concerned are derivatives of indole and carbazole and are the second reported series of non-competitive antagonists of the GluK2 receptor (the first on...
Autores principales: | Kaczor, Agnieszka A., Wróbel, Tomasz, Kronbach, Christiane, Unverferth, Klaus, Stachal, Tomasz, Matosiuk, Dariusz |
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Formato: | Online Artículo Texto |
Lenguaje: | English |
Publicado: |
Springer US
2014
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Materias: | |
Acceso en línea: | https://www.ncbi.nlm.nih.gov/pmc/articles/PMC4295030/ https://www.ncbi.nlm.nih.gov/pubmed/25620864 http://dx.doi.org/10.1007/s00044-014-1171-1 |
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