Cargando…

Novel heteroaryl phosphonicdiamides PTPs inhibitors as anti-hyperglycemic agents

BACKGROUND: Chronic and oral administration of benzylamine improves glucose tolerance. Picolylamine is a selective functional antagonist of the human adenosine A(2B) receptor. Phosphonic diamide derivatives enhance the cellular permeability and in turn their biological activities. METHODS: A series...

Descripción completa

Detalles Bibliográficos
Autores principales:	Sekhar, Kuruva Chandra, Syed, Rasheed, Golla, Madhava, MV, Jyothi Kumar, Yellapu, Nanda Kumar, Chippada, Appa Rao, Chamarthi, Naga Raju
Formato:	Online Artículo Texto
Lenguaje:	English
Publicado:	BioMed Central 2014
Materias:	Research Article
Acceso en línea:	https://www.ncbi.nlm.nih.gov/pmc/articles/PMC4305230/ https://www.ncbi.nlm.nih.gov/pubmed/25542373 http://dx.doi.org/10.1186/s40199-014-0076-3

Ejemplares similares

Molecular designing and in silico evaluation of darunavir derivatives as anticancer agents
por: Mahto, Manoj kumar, et al.
Publicado: (2014)

Development of a pronunciation teaching perception scale (PTPS) for preservice English language teachers
por: Ercan, Halil, et al.
Publicado: (2022)

Antidiabetic and antihyperlipidemic activity of Piper longum root aqueous extract in STZ induced diabetic rats
por: Nabi, Shaik Abdul, et al.
Publicado: (2013)

Disruption of PTPS Gene Causing Pale Body Color and Lethal Phenotype in the Silkworm, Bombyx mori
por: Tong, Xiaoling, et al.
Publicado: (2018)

Construction, Factor Structure, and Internal Consistency Reliability of the Hospital Physical Therapy Perceived Satisfaction Questionnaire (H-PTPS)
por: Albornoz-Cabello, Manuel, et al.
Publicado: (2020)

New Urea and Thiourea Derivatives of Piperazine Doped with Febuxostat: Synthesis and Evaluation of Anti-TMV and Antimicrobial Activities
por: Krishna Reddy, Reddivari Chenna, et al.
Publicado: (2013)

Arylation and Heteroarylation of Thienylsulfonamides with Organotrifluoroborates
por: Noreen, Mnaza, et al.
Publicado: (2014)

Exosome-driven transfer of tumor-associated Pioneer Translation Products (TA-PTPs) for the MHC class I cross-presentation pathway
por: Duvallet, Emilie, et al.
Publicado: (2016)

Performance of the Southend pre-test probability score (PTPS) for giant cell arteritis in a fast-track clinic in Western Australia
por: Mathake, Mmoloki, et al.
Publicado: (2022)

Enzymatic Enantioselective Decarboxylative Protonation of Heteroaryl Malonates
por: Lewin, Ross, et al.
Publicado: (2015)

Palladium-catalysed synthesis of triaryl(heteroaryl)methanes
por: Zhang, Shuguang, et al.
Publicado: (2017)

Heteroaryl Chalcones: Design, Synthesis, X-ray Crystal Structures and Biological Evaluation
por: Kumar, C. S. Chidan, et al.
Publicado: (2013)

Deoxygenative C2-heteroarylation of quinoline N-oxides: facile access to α-triazolylquinolines
por: Sontakke, Geetanjali S, et al.
Publicado: (2021)

Modeling, molecular docking, probing catalytic binding mode of acetyl-CoA malate synthase G in Brucella melitensis 16M
por: Adi, Pradeepkiran Jangampalli, et al.
Publicado: (2016)

Palladium-catalyzed difluoromethylation of heteroaryl chlorides, bromides and iodides
por: Lu, Changhui, et al.
Publicado: (2017)

Redox-enabled direct stereoconvergent heteroarylation of simple alcohols
por: Liu, Yongbing, et al.
Publicado: (2021)

Central Diabetes Insipidus and Hyperglycemic Hyperosmolar State Following Accidental Carbon Monoxide Poisoning
por: Ul Abideen, Zain, et al.
Publicado: (2017)

Modeling, molecular dynamics, and docking assessment of transcription factor rho: a potential drug target in Brucella melitensis 16M
por: Pradeepkiran, Jangampalli Adi, et al.
Publicado: (2015)

One-Pot Synthesis and Applications of N-Heteroaryl Iodonium Salts
por: Bielawski, Marcin, et al.
Publicado: (2014)

A practical and scalable system for heteroaryl amino acid synthesis
por: Aycock, R. A., et al.
Publicado: (2017)

Direct heteroarylation polymerization: guidelines for defect-free conjugated polymers
por: Bura, Thomas, et al.
Publicado: (2017)

Chemospecific Cyclizations of α‐Carbonyl Sulfoxonium Ylides on Aryls and Heteroaryls
por: Clare, Daniel, et al.
Publicado: (2019)

Synthesis of Bis-heteroaryls Using Grignard Reagents and Pyridylsulfonium Salts
por: Horan, Alexandra M., et al.
Publicado: (2021)

Synthesis and evaluation of new heteroaryl nitrones with spin trap properties
por: Barriga-González, G., et al.
Publicado: (2020)

Synthesis, in vitro bioassays, and computational study of heteroaryl nitazoxanide analogs
por: Ahmed, Tasmia, et al.
Publicado: (2021)

Catalyst-free assembly of giant tris(heteroaryl)methanes: synthesis of novel pharmacophoric triads and model sterically crowded tris(heteroaryl/aryl)methyl cation salts
por: Abonia, Rodrigo, et al.
Publicado: (2019)

Conformational transition pathway of R308K mutant glucokinase in the presence of the glucokinase activator YNKGKA4
por: Yellapu, Nanda Kumar, et al.
Publicado: (2018)

Synthesis of novel 5-alkyl/aryl/heteroaryl substituted diethyl 3,4-dihydro-2H-pyrrole-4,4-dicarboxylates by aziridine ring expansion of 2-[(aziridin-1-yl)-1-alkyl/aryl/heteroaryl-methylene]malonic acid diethyl esters
por: More, Satish S, et al.
Publicado: (2011)

Anti-hyperglycemic activity of Caralluma umbellata Haw.
por: Bellamakondi, Pavan Kumar, et al.
Publicado: (2014)

Hyperglycemic chorea
por: Sasaki, Tokio, et al.
Publicado: (2021)

Prospects to the formation and control of potential dimer impurity E of pantoprazole sodium sesquihydrate
por: Awasthi, Arun Kumar, et al.
Publicado: (2019)

Fluorescent hexaaryl- and hexa-heteroaryl[3]radialenes: Synthesis, structures, and properties
por: Avellaneda, Antonio, et al.
Publicado: (2012)

Amination of Heteroaryl Chlorides: Palladium Catalysis or S(N)Ar in Green Solvents?
por: Walsh, Katie, et al.
Publicado: (2013)

Copper-Mediated Perfluoroalkylation of Heteroaryl Bromides with (phen)CuR(F)
por: Mormino, Michael G., et al.
Publicado: (2014)

In-Depth Assessment of the Palladium-Catalyzed Fluorination of Five-Membered Heteroaryl Bromides
por: Milner, Phillip J., et al.
Publicado: (2015)

Palladium-catalyzed difluoromethylthiolation of heteroaryl bromides, iodides, triflates and aryl iodides
por: Wu, Jiang, et al.
Publicado: (2016)

Synthesis of Novel Aryl(heteroaryl)sulfonyl Ureas of Possible Biological Interest
por: Sączewski, Franciszek, et al.
Publicado: (2010)

Antitumoural Sulphur and Selenium Heteroaryl Compounds: Thermal Characterization and Stability Evaluation
por: Alcolea, Verónica, et al.
Publicado: (2017)

Organocatalyzed, Photoredox Heteroarylation of 2-Trifluoroboratochromanones via C–H Functionalization
por: Matsui, Jennifer K., et al.
Publicado: (2017)

Investigation on the Synthesis, Application and Structural Features of Heteroaryl 1,2-Diketones
por: Wehrle, Robert J., et al.
Publicado: (2022)

Cannot write session to /tmp/vufind_sessions/sess_37r948fmcseiatvbuq5bbqfo3a