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Efficient Regioselective Ring Opening of Activated Aziridine-2-Carboxylates with [(18)F]Fluoride

Aziridines can undergo a range of ring-opening reactions with nucleophiles. The regio- and stereochemistry of the products depend on the substituents on the aziridine. Aziridine ring-opening reactions have rarely been used in radiosynthesis. Herein we report the ring opening of activated aziridine-2...

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Detalles Bibliográficos
Autores principales:	Schjoeth-Eskesen, Christina, Hansen, Paul Robert, Kjaer, Andreas, Gillings, Nic
Formato:	Online Artículo Texto
Lenguaje:	English
Publicado:	BlackWell Publishing Ltd 2015
Materias:	Full Papers
Acceso en línea:	https://www.ncbi.nlm.nih.gov/pmc/articles/PMC4380955/ https://www.ncbi.nlm.nih.gov/pubmed/25861572 http://dx.doi.org/10.1002/open.201402081

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