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3-Glucosylated 5-amino-1,2,4-oxadiazoles: synthesis and evaluation as glycogen phosphorylase inhibitors

Glycogen phosporylase (GP) is a promising target for the control of glycaemia. The design of inhibitors binding at the catalytic site has been accomplished through various families of glucose-based derivatives such as oxadiazoles. Further elaboration of the oxadiazole aromatic aglycon moiety is now...

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Detalles Bibliográficos
Autores principales:	Donnier-Maréchal, Marion, Goyard, David, Folliard, Vincent, Docsa, Tibor, Gergely, Pal, Praly, Jean-Pierre, Vidal, Sébastien
Formato:	Online Artículo Texto
Lenguaje:	English
Publicado:	Beilstein-Institut 2015
Materias:	Full Research Paper
Acceso en línea:	https://www.ncbi.nlm.nih.gov/pmc/articles/PMC4419504/ https://www.ncbi.nlm.nih.gov/pubmed/25977724 http://dx.doi.org/10.3762/bjoc.11.56

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