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Design and Synthesis of Novel N-Arylsulfonyl-3-(2-yl-ethanone)-6-methylindole Derivatives as Inhibitors of HIV-1 Replication

Seven novel N-arylsulfonyl-3-(2-yl-ethanone)-6-methylindole derivatives 4a–f and 6 were readily synthesized and have been identified as inhibitors of human immunodeficiency virus type-1 (HIV-1) replication. Initial biological studies indicated that among these derivatives, N-(p-ethyl)phenylsulfonyl-...

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Detalles Bibliográficos
Autores principales:	Che, Zhiping, Liu, Shengming, Tian, Yuee, Hu, Zhenjie, Chen, Yingwu, Chen, Genqiang
Formato:	Online Artículo Texto
Lenguaje:	English
Publicado:	MDPI 2015
Materias:	Article
Acceso en línea:	https://www.ncbi.nlm.nih.gov/pmc/articles/PMC4491657/ https://www.ncbi.nlm.nih.gov/pubmed/26110320 http://dx.doi.org/10.3390/ph8020221

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