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2-acetylphenol analogs as potent reversible monoamine oxidase inhibitors
Based on a previous report that substituted 2-acetylphenols may be promising leads for the design of novel monoamine oxidase (MAO) inhibitors, a series of C5-substituted 2-acetylphenol analogs (15) and related compounds (two) were synthesized and evaluated as inhibitors of human MAO-A and MAO-B. Gen...
Autores principales: | Legoabe, Lesetja J, Petzer, Anél, Petzer, Jacobus P |
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Formato: | Online Artículo Texto |
Lenguaje: | English |
Publicado: |
Dove Medical Press
2015
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Materias: | |
Acceso en línea: | https://www.ncbi.nlm.nih.gov/pmc/articles/PMC4507791/ https://www.ncbi.nlm.nih.gov/pubmed/26203229 http://dx.doi.org/10.2147/DDDT.S86225 |
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