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A calixpyrrole derivative acts as an antagonist to GPER, a G-protein coupled receptor: mechanisms and models

Estrogens regulate numerous pathophysiological processes, mainly by binding to and activating estrogen receptor (ER)α and ERβ. Increasing amounts of evidence have recently demonstrated that G-protein coupled receptor 30 (GPR30; also known as GPER) is also involved in diverse biological responses to...

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Detalles Bibliográficos
Autores principales:	Lappano, Rosamaria, Rosano, Camillo, Pisano, Assunta, Santolla, Maria Francesca, De Francesco, Ernestina Marianna, De Marco, Paola, Dolce, Vincenza, Ponassi, Marco, Felli, Lamberto, Cafeo, Grazia, Kohnke, Franz Heinrich, Abonante, Sergio, Maggiolini, Marcello
Formato:	Online Artículo Texto
Lenguaje:	English
Publicado:	The Company of Biologists 2015
Materias:	Research Article
Acceso en línea:	https://www.ncbi.nlm.nih.gov/pmc/articles/PMC4610237/ https://www.ncbi.nlm.nih.gov/pubmed/26183213 http://dx.doi.org/10.1242/dmm.021071

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