Cargando…

Synthesis of constrained analogues of tryptophan

A Lewis acid-catalysed diastereoselective [4 + 2] cycloaddition of vinylindoles and methyl 2-acetamidoacrylate, leading to methyl 3-acetamido-1,2,3,4-tetrahydrocarbazole-3-carboxylate derivatives, is described. Treatment of the obtained cycloadducts under hydrolytic conditions results in the prepara...

Descripción completa

Detalles Bibliográficos
Autores principales:	Rossi, Elisabetta, Pirovano, Valentina, Negrato, Marco, Abbiati, Giorgio, Dell’Acqua, Monica
Formato:	Online Artículo Texto
Lenguaje:	English
Publicado:	Beilstein-Institut 2015
Materias:	Full Research Paper
Acceso en línea:	https://www.ncbi.nlm.nih.gov/pmc/articles/PMC4661003/ https://www.ncbi.nlm.nih.gov/pubmed/26664620 http://dx.doi.org/10.3762/bjoc.11.216

Ejemplares similares

Synthesis of Cyclohepta[b]indoles by (4 + 3) Cycloaddition of 2-Vinylindoles or 4H-Furo[3,2-b]indoles with Oxyallyl Cations
por: Pirovano, Valentina, et al.
Publicado: (2020)

Side Chain Orientation of Tryptophan Analogues Determines Agonism and Inverse Agonism in Short Ghrelin Peptides
por: Nicke, Lennart, et al.
Publicado: (2019)

Synthesis and Biological Evaluation of New (−)‐Englerin Analogues
por: López‐Suárez, Laura, et al.
Publicado: (2016)

Enantiospecific Synthesis and Cytotoxicity Evaluation of Oximidine II Analogues
por: Schneider, Christopher M., et al.
Publicado: (2016)

Synthesis of gem-difluoromethylenated analogues of boronolide
por: Lin, Jing, et al.
Publicado: (2010)

An improved synthesis of adefovir and related analogues
por: Jones, David J, et al.
Publicado: (2019)

Synthesis and Biological Evaluation of Dantrolene‐Like Hydrazide and Hydrazone Analogues as Multitarget Agents for Neurodegenerative Diseases
por: Bolognino, Isabella, et al.
Publicado: (2021)

Synthesis of phosphonate and phostone analogues of ribose-1-phosphates
por: Nasomjai, Pitak, et al.
Publicado: (2009)

Synthesis of some novel hydrazono acyclic nucleoside analogues
por: Soltani Rad, Mohammad N, et al.
Publicado: (2010)

Synthesis of 4” manipulated Lewis X trisaccharide analogues
por: Moore, Christopher J, et al.
Publicado: (2012)

A chemoselective and continuous synthesis of m-sulfamoylbenzamide analogues
por: Verlee, Arno, et al.
Publicado: (2017)

Synthesis of ribavirin 2’-Me-C-nucleoside analogues
por: Cosson, Fanny, et al.
Publicado: (2017)

Synthesis of 2-substituted tryptophans via a C3- to C2-alkyl migration
por: Mari, Michele, et al.
Publicado: (2014)

Anti‐flavivirus Activity of Different Tritylated Pyrimidine and Purine Nucleoside Analogues
por: McGuigan, Christopher, et al.
Publicado: (2016)

Synthesis of crispine A analogues via an intramolecular Schmidt reaction
por: Kapat, Ajoy, et al.
Publicado: (2007)

Synthesis and conformational preferences of short analogues of antifreeze glycopeptides (AFGP)
por: Urbańczyk, Małgorzata, et al.
Publicado: (2019)

Efficient synthesis of dipeptide analogues of α-fluorinated β-aminophosphonates
por: Kaźmierczak, Marcin, et al.
Publicado: (2020)

Synthesis of novel sulfide-based cyclic peptidomimetic analogues to solonamides
por: Brango-Vanegas, José, et al.
Publicado: (2019)

Towards Photochromic Azobenzene‐Based Inhibitors for Tryptophan Synthase
por: Simeth, Nadja A., et al.
Publicado: (2020)

Heck Diversification of Indole‐Based Substrates under Aqueous Conditions: From Indoles to Unprotected Halo‐tryptophans and Halo‐tryptophans in Natural Product Derivatives
por: Pubill‐Ulldemolins, Cristina, et al.
Publicado: (2019)

Total Synthesis of Viniferifuran, Resveratrol‐Piceatannol Hybrid, Anigopreissin A and Analogues – Investigation of Demethylation Strategies
por: Vo, Duc Duy, et al.
Publicado: (2016)

Synthesis and Cell Growth Inhibitory Activity of Six Non‐glycosaminoglycan‐Type Heparin‐Analogue Trisaccharides
por: Lisztes, Erika, et al.
Publicado: (2021)

Synthesis of (−)-julocrotine and a diversity oriented Ugi-approach to analogues and probes
por: Neves Filho, Ricardo A W, et al.
Publicado: (2011)

Synthesis and antiviral activities of spacer-linked 1-thioglucuronide analogues of glycyrrhizin
por: Stanetty, Christian, et al.
Publicado: (2012)

Gold(I)-catalysed synthesis of a furan analogue of thiamine pyrophosphate
por: Iqbal, Amjid, et al.
Publicado: (2014)

Design and synthesis of diazine-based panobinostat analogues for HDAC8 inhibition
por: Balasubramaniam, Sivaraman, et al.
Publicado: (2020)

Silver and gold-catalyzed multicomponent reactions
por: Abbiati, Giorgio, et al.
Publicado: (2014)

Synthesis of thienyl analogues of PCBM and investigation of morphology of mixtures in P3HT
por: Matsumoto, Fukashi, et al.
Publicado: (2008)

Synthesis of a new class of aminocyclitol analogues with the conduramine D-2 configuration
por: Kelebekli, Latif, et al.
Publicado: (2010)

Synthesis of pyrrolidine-based hamamelitannin analogues as quorum sensing inhibitors in Staphylococcus aureus
por: Bouton, Jakob, et al.
Publicado: (2018)

Incorporation of tryptophan analogues into the lantibiotic nisin
por: Zhou, Liang, et al.
Publicado: (2016)

Synthesis of Hollow Co–Fe Prussian Blue Analogue Cubes by using Silica Spheres as a Sacrificial Template
por: Azhar, Alowasheeir, et al.
Publicado: (2018)

Synthesis and Cytotoxicity Evaluation of C4‐ and C5‐Modified Analogues of the α,β‐Unsaturated Lactone of Pironetin
por: Huang, David S., et al.
Publicado: (2017)

The multicomponent approach to N-methyl peptides: total synthesis of antibacterial (–)-viridic acid and analogues
por: Neves Filho, Ricardo A W, et al.
Publicado: (2012)

Diastereoselective synthesis of new O-alkylated and C-branched inositols and their corresponding fluoro analogues
por: Collet, Charlotte, et al.
Publicado: (2016)

Semi-synthesis and insecticidal activity of spinetoram J and its D-forosamine replacement analogues
por: Zhang, Kai, et al.
Publicado: (2018)

Revaluation of biomass-derived furfuryl alcohol derivatives for the synthesis of carbocyclic nucleoside phosphonate analogues
por: Sidi Mohamed, Bemba, et al.
Publicado: (2017)

Enantiomerically Pure Constrained Geometry Complexes of the Rare‐Earth Metals Featuring a Dianionic N‐Donor Functionalised Pentadienyl Ligand: Synthesis and Characterisation
por: Münster, Katharina, et al.
Publicado: (2020)

Solid‐Phase Synthesis of Fluorinated Analogues of Glycosyl 1‐Phosphate Repeating Structures from Leishmania using the Phosphoramidite Method
por: Hara, Rintaro Iwata, et al.
Publicado: (2018)

A new method for the synthesis of α-aminoalkylidenebisphosphonates and their asymmetric phosphonyl-phosphinyl and phosphonyl-phosphinoyl analogues
por: Kuźnik, Anna, et al.
Publicado: (2015)

Cannot write session to /tmp/vufind_sessions/sess_bhjq92tcda9dcvoc708oudftbj