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Synthesis of [(18)F]Arenes via the Copper-Mediated [(18)F]Fluorination of Boronic Acids

[Image: see text] A copper-mediated radiofluorination of aryl- and vinylboronic acids with K(18)F is described. This method exhibits high functional group tolerance and is effective for the radiofluorination of a range of electron-deficient, -neutral, and -rich aryl-, heteroaryl-, and vinylboronic a...

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Detalles Bibliográficos
Autores principales:	Mossine, Andrew V., Brooks, Allen F., Makaravage, Katarina J., Miller, Jason M., Ichiishi, Naoko, Sanford, Melanie S., Scott, Peter J. H.
Formato:	Online Artículo Texto
Lenguaje:	English
Publicado:	American Chemical Society 2015
Acceso en línea:	https://www.ncbi.nlm.nih.gov/pmc/articles/PMC4672358/ https://www.ncbi.nlm.nih.gov/pubmed/26568457 http://dx.doi.org/10.1021/acs.orglett.5b02875

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