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Synthesis and Biological Activity of New [1,3]Thiazolo[4,5-d]pyridazin-4(5H)-ones

A series of novel 2-(N-pyrrolidino, N-piperidino or N-morpholino)-7-phenyl(α-furoyl or α-thienyl)-[1,3]thiazolo[4,5-d]pyridazinones 10a–c, 14–16a,b was synthesized in 78–87% yields via the reaction of methyl 5-benzoyl(α-furoyl or α-thienyl)-2-aminosubstituted-thiazol-4-carboxylates 9a–c, 13a–e with...

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Detalles Bibliográficos
Autores principales:	Demchenko, Anatoly, Bobkova, Ludmila, Yadlovskiy, Oleh, Buchtiarova, Tatiana, Demchenko, Sergey
Formato:	Online Artículo Texto
Lenguaje:	English
Publicado:	The Austrian Journal of Pharmaceutical Sciences 2016
Materias:	Research Article
Acceso en línea:	https://www.ncbi.nlm.nih.gov/pmc/articles/PMC4871179/ https://www.ncbi.nlm.nih.gov/pubmed/27222602 http://dx.doi.org/10.3797/scipharm.1505-16

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