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Synthesis and Biological Evaluation of New (−)‐Englerin Analogues

We report the synthesis and biological evaluation of a series of (−)‐englerin A analogues obtained along our previously reported synthetic route based on a stereoselective gold(I) cycloaddition process. This synthetic route is a convenient platform to access analogues with broad structural diversity...

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Detalles Bibliográficos
Autores principales:	López‐Suárez, Laura, Riesgo, Lorena, Bravo, Fernando, Ransom, Tanya T., Beutler, John A., Echavarren, Antonio M.
Formato:	Online Artículo Texto
Lenguaje:	English
Publicado:	John Wiley and Sons Inc. 2016
Materias:	Full Papers
Acceso en línea:	https://www.ncbi.nlm.nih.gov/pmc/articles/PMC4926265/ https://www.ncbi.nlm.nih.gov/pubmed/27005578 http://dx.doi.org/10.1002/cmdc.201600040

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