Cargando…

Role of fosaprepitant, a neurokinin Type 1 receptor antagonist, in morphine-induced antinociception in rats

OBJECTIVES: Opioids such as morphine form the cornerstone in the treatment of moderate to severe pain. However, opioids also produce serious side effects such as tolerance. Fosaprepitant is a substance P (SP) receptor antagonist, which is used for treating chemotherapy-induced nausea and vomiting. S...

Descripción completa

Detalles Bibliográficos
Autores principales:	Prasoon, Pranav, Gupta, Shivani, Kumar, Rahul, Gautam, Mayank, Kaler, Saroj, Ray, Subrata Basu
Formato:	Online Artículo Texto
Lenguaje:	English
Publicado:	Medknow Publications & Media Pvt Ltd 2016
Materias:	Research Article
Acceso en línea:	https://www.ncbi.nlm.nih.gov/pmc/articles/PMC4980927/ https://www.ncbi.nlm.nih.gov/pubmed/27756950 http://dx.doi.org/10.4103/0253-7613.186198

Ejemplares similares

Comparative antinociceptive effect of arachidonylcyclopropylamide, a cannabinoid 1 receptor agonist & lignocaine, a local anaesthetic agent, following direct intrawound administration in rats
por: Kumar, Rahul, et al.
Publicado: (2016)

Diverse characters of Brennan’s paw incision model regarding certain parameters in the rat
por: Kumar, Rahul, et al.
Publicado: (2019)

Comparison of Antinociceptive Effect of Octreotide With Morphine in a Rat Model of Acute Inflammatory Pain
por: Singh, Perminder, et al.
Publicado: (2021)

Evaluation of the Antinociceptive Effect of Maropitant, a Neurokinin-1 Receptor Antagonist, in Cats Undergoing Ovariohysterectomy
por: Corrêa, Janaina M. X., et al.
Publicado: (2019)

Nimodipine potentiates the analgesic effect of morphine in the rat hot-plate test: Implications in the treatment of pain
por: Kumar, Rakesh, et al.
Publicado: (2011)

Neurokinin 1 Receptor Antagonists for Pruritus
por: Alam, Majid, et al.
Publicado: (2021)

Neurokinin-1 Receptor Antagonists against Hepatoblastoma
por: Muñoz, Miguel, et al.
Publicado: (2019)

In vivo antinociception of potent mu opioid agonist tetrapeptide analogues and comparison with a compact opioid agonist - neurokinin 1 receptor antagonist chimera
por: Guillemyn, Karel, et al.
Publicado: (2012)

Central and peripheral relationships between morphine and glucose on antinociception in rats
por: Yamamoto, Rinah T., et al.
Publicado: (2014)

A Comparison of the Antinociceptive Properties of SJP-005 and Morphine in Rats
por: Verster, Joris C, et al.
Publicado: (2021)

Intrathecal Catheterization and Drug Delivery in Rats to Compare the Analgesic Effects of Morphine with Ketorolac
por: Ray, Subrata Basu, et al.
Publicado: (2011)

Long-term Morphine-treated Rats are more Sensitive to Antinociceptive Effect of Diclofenac than the Morphine-naive rats
por: Akbari, Esmaeil, et al.
Publicado: (2013)

Effect of Nimodipine on Morphine-related Withdrawal Syndrome in Rat Model: An Observational Study
por: Mishra, Pravash Ranjan, et al.
Publicado: (2017)

Additive Antinociception between Intrathecal Sildenafil and Morphine in the Rat Formalin Test
por: Yoon, Myung Ha, et al.
Publicado: (2008)

Antinociceptive Effect of Memantine and Morphine on Vincristine-induced Peripheral Neuropathy in Rats
por: Park, Byoung Yoon, et al.
Publicado: (2010)

Data on prolonged morphine-induced antinociception and behavioral inhibition in older rats
por: Paul, Alok Kumar, et al.
Publicado: (2018)

Intrathecal Co-administration of Morphine Facilitated the Anti-nociceptive of Bupivacaine in a Rat Model of Acute Postoperative Pain
por: Ghosh, Tamoghna, et al.
Publicado: (2022)

Treating hot flushes with a neurokinin 3 receptor antagonist
por: Prague, Julia K., et al.
Publicado: (2017)

Neurokinin 3 receptor antagonists for menopausal vasomotor symptoms, an appraisal
por: Gompel, Anne, et al.
Publicado: (2023)

Neurokinin Receptor Antagonist, Fezolinetant, for Treatment of Menopausal Vasomotor Symptoms
por: Pinkerton, JoAnn V, et al.
Publicado: (2023)

Intrathecal Lamotrigine Attenuates Antinociceptive Morphine Tolerance and Suppresses Spinal Glial Cell Activation in Morphine-Tolerant Rats
por: Jun, In-Gu, et al.
Publicado: (2013)

Selective antinociceptive effects of a combination of the N-methyl-D-aspartate receptor peptide antagonist [Ser(1)]histogranin and morphine in rat models of pain
por: Hama, Aldric, et al.
Publicado: (2014)

Morphine Antinociception Restored by Use of Methadone in the Morphine-Resistant Inflammatory Pain State
por: Watanabe, Chizuko, et al.
Publicado: (2020)

Antinociceptive Effect of Intrathecal Nefopam and Interaction with Morphine in Formalin-Induced Pain of Rats
por: Cho, Soo Young, et al.
Publicado: (2013)

Effects of an intrathecal TRPV1 antagonist, SB366791, on morphine-induced itch, body temperature, and antinociception in mice
por: Sakakibara, Satoshi, et al.
Publicado: (2019)

Neurokinin-1 Receptor Antagonist Treatment in Polymicrobial Sepsis: Molecular Insights
por: Hegde, Akhil, et al.
Publicado: (2010)

Neurokinin-1 receptor antagonists: A new revolution in antiretroviral treatment?
por: Grewal, Udhayvir Singh
Publicado: (2016)

The Neurokinin-1 Receptor Antagonist Aprepitant: An Intelligent Bullet against Cancer?
por: Muñoz, Miguel, et al.
Publicado: (2020)

Zimelidine attenuates the development of tolerance to morphine-induced antinociception
por: Ozdemir, Ercan, et al.
Publicado: (2012)

Exercise Reduces Morphine-Induced Hyperalgesia and Antinociceptive Tolerance
por: Gong, Xingrui, et al.
Publicado: (2021)

Differences in morphine-induced antinociception in male and female offspring born of morphine exposed mothers
por: Biglarnia, Masoomeh, et al.
Publicado: (2013)

Functionally Selective Signaling for Morphine and Fentanyl Antinociception and Tolerance Mediated by the Rat Periaqueductal Gray
por: Morgan, Michael M., et al.
Publicado: (2014)

Antiemetic Prophylaxis with Fosaprepitant and 5-HT(3)-Receptor Antagonists in Pediatric Patients Undergoing Autologous Hematopoietic Stem Cell Transplantation
por: Cabanillas Stanchi, Karin Melanie, et al.
Publicado: (2020)

Study of antinociceptive activity of SSRI (fluoxetine and escitalopram) and atypical antidepressants (venlafaxine and mirtazepine) and their interaction with morphine and naloxone in mice
por: Sikka, Pranav, et al.
Publicado: (2011)

The Neurokinin 1 Receptor Antagonist, Ezlopitant, Reduces Appetitive Responding for Sucrose and Ethanol
por: Steensland, Pia, et al.
Publicado: (2010)

Evolving role of neurokinin 1-receptor antagonists for chemotherapy-induced nausea and vomiting
por: Navari, Rudolph M, et al.
Publicado: (2018)

Crystal structures of the human neurokinin 1 receptor in complex with clinically used antagonists
por: Schöppe, Jendrik, et al.
Publicado: (2019)

Neurokinin receptor antagonists as potential non-hormonal treatments for vasomotor symptoms of menopause
por: Conklin, Melissa, et al.
Publicado: (2023)

The effect of gut microbiome on tolerance to morphine mediated antinociception in mice
por: Kang, Minho, et al.
Publicado: (2017)

Enhancement of morphine-induced antinociception after electroconvulsive shock in mice
por: Iwata, Ken, et al.
Publicado: (2021)

Cannot write session to /tmp/vufind_sessions/sess_kknba6j9e02e9oh13fdusclakp