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In Vitro Metabolic Studies of REV-ERB Agonists SR9009 and SR9011

SR9009 and SR9011 are attractive as performance-enhancing substances due to their REV-ERB agonist effects and thus circadian rhythm modulation activity. Although no pharmaceutical preparations are available yet, illicit use of SR9009 and SR9011 for doping purposes can be anticipated, especially sinc...

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Detalles Bibliográficos
Autores principales:	Geldof, Lore, Deventer, Koen, Roels, Kris, Tudela, Eva, Van Eenoo, Peter
Formato:	Online Artículo Texto
Lenguaje:	English
Publicado:	MDPI 2016
Materias:	Article
Acceso en línea:	https://www.ncbi.nlm.nih.gov/pmc/articles/PMC5085709/ https://www.ncbi.nlm.nih.gov/pubmed/27706103 http://dx.doi.org/10.3390/ijms17101676

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