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Synthesis of 2-tetrafluoropyridyl-4,5-disubstituted 1,2,3-triazoles

ABSTRACT: By cycloaddition reaction of sodium azide with chalcone in the presence of CuO as a catalyst in DMF a 1,2,3-triazole are prepared in reaction with pentafluoropyridine to give 2-(tetrafluoropyridin-4-yl)-1,2,3-triazole derivatives in good yields and high regioselectivity. The regioselectivi...

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Detalles Bibliográficos
Autores principales:	Beyki, Khalil, Maghsoodlou, Malek Taher, Heydari, Reza
Formato:	Online Artículo Texto
Lenguaje:	English
Publicado:	Springer International Publishing 2016
Materias:	Short Report
Acceso en línea:	https://www.ncbi.nlm.nih.gov/pmc/articles/PMC5106409/ https://www.ncbi.nlm.nih.gov/pubmed/27933240 http://dx.doi.org/10.1186/s40064-016-3398-4

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