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Ciproxifan, a histamine H(3) receptor antagonist, reversibly inhibits monoamine oxidase A and B
Ciproxifan is a well-investigated histamine H(3) receptor (H3R) inverse agonist/antagonist, showing an exclusively high species-specific affinity at rodent compared to human H3R. It is well studied as reference compound for H3R in rodent models for neurological diseases connected with neurotransmitt...
Autores principales: | Hagenow, S., Stasiak, A., Ramsay, R. R., Stark, H. |
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Formato: | Online Artículo Texto |
Lenguaje: | English |
Publicado: |
Nature Publishing Group
2017
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Materias: | |
Acceso en línea: | https://www.ncbi.nlm.nih.gov/pmc/articles/PMC5233962/ https://www.ncbi.nlm.nih.gov/pubmed/28084411 http://dx.doi.org/10.1038/srep40541 |
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