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cis-Diastereoselective synthesis of chroman-fused tetralins as B-ring-modified analogues of brazilin

We have synthesized a series of cis-6a,7,8,12b-tetrahydro-6H-naphtho[2,1-c]chromen-6a-ols as B-ring-modified analogues of (±)-brazilin. A completely regio- and cis-diastereoselective intramolecular Friedel–Crafts epoxy–arene cyclization of 1-tetralone-derived glycidyl ethers catalyzed by Brønsted ac...

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Detalles Bibliográficos
Autores principales:	Gogoi, Dimpee, Devi, Runjun, Pahari, Pallab, Sarma, Bipul, Das, Sajal Kumar
Formato:	Online Artículo Texto
Lenguaje:	English
Publicado:	Beilstein-Institut 2016
Materias:	Letter
Acceso en línea:	https://www.ncbi.nlm.nih.gov/pmc/articles/PMC5238543/ https://www.ncbi.nlm.nih.gov/pubmed/28144354 http://dx.doi.org/10.3762/bjoc.12.280

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