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New Synthesis, Structure and Analgesic Properties of Methyl 1-R-4-Methyl-2,2-Dioxo-1H-2λ(6),1-Benzothiazine-3-Carboxylates

According to the principles of the methodology of bioisosteric replacements a series of methyl 1-R-4-methyl-2,2-dioxo-1H-2λ(6),1-benzothiazine-3-carboxylates has been obtained as potential analgesics. In addition, a fundamentally new strategy for the synthesis of compounds of this chemical class inv...

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Detalles Bibliográficos
Autores principales:	Azotla-Cruz, Liliana, Lijanova, Irina V., Ukrainets, Igor V., Likhanova, Natalya V., Olivares-Xometl, Octavio, Bereznyakova, Natalya L.
Formato:	Online Artículo Texto
Lenguaje:	English
Publicado:	MDPI 2017
Materias:	Article
Acceso en línea:	https://www.ncbi.nlm.nih.gov/pmc/articles/PMC5388141/ https://www.ncbi.nlm.nih.gov/pubmed/28085092 http://dx.doi.org/10.3390/scipharm85010002

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