Cargando…
New MT(2) Melatonin Receptor-Selective Ligands: Agonists and Partial Agonists
The search for melatonin receptor agonists and antagonists specific towards one of the receptor subtypes will extend our understanding of the role of this system in relaying circadian information to the body. A series of compounds derived from a hit compound discovered in a screening process led to...
Autores principales: | Boutin, Jean A., Bonnaud, Anne, Brasseur, Chantal, Bruno, Olivier, Lepretre, Nolwenn, Oosting, Peter, Coumailleau, Sophie, Delagrange, Philippe, Nosjean, Olivier, Legros, Céline |
---|---|
Formato: | Online Artículo Texto |
Lenguaje: | English |
Publicado: |
MDPI
2017
|
Materias: | |
Acceso en línea: | https://www.ncbi.nlm.nih.gov/pmc/articles/PMC5535840/ https://www.ncbi.nlm.nih.gov/pubmed/28644418 http://dx.doi.org/10.3390/ijms18071347 |
Ejemplares similares
-
Characterization of the various functional pathways elicited by synthetic agonists or antagonists at the melatonin MT(1) and MT(2) receptors
por: Legros, Céline, et al.
Publicado: (2019) -
Hamster Melatonin Receptors: Cloning and Binding Characterization of MT(1) and Attempt to Clone MT(2)
por: Gautier, Célia, et al.
Publicado: (2018) -
Recombinant Human Melatonin Receptor MT1 Isolated in Mixed Detergents Shows Pharmacology Similar to That in Mammalian Cell Membranes
por: Logez, Christel, et al.
Publicado: (2014) -
New Radioligands for Describing the Molecular Pharmacology of MT(1) and MT(2) Melatonin Receptors
por: Legros, Céline, et al.
Publicado: (2013) -
Structural Basis for Agonistic Activity and Selectivity toward Melatonin Receptors hMT1 and hMT2
por: Cantarini, Mattia, et al.
Publicado: (2023)