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Azemiopsin, a Selective Peptide Antagonist of Muscle Nicotinic Acetylcholine Receptor: Preclinical Evaluation as a Local Muscle Relaxant

Azemiopsin (Az), a linear peptide from the Azemiops feae viper venom, contains no disulfide bonds, is a high-affinity and selective inhibitor of nicotinic acetylcholine receptor (nAChR) of muscle type and may be considered as potentially applicable nondepolarizing muscle relaxant. In this study, we...

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Detalles Bibliográficos
Autores principales:	Shelukhina, Irina V., Zhmak, Maxim N., Lobanov, Alexander V., Ivanov, Igor A., Garifulina, Alexandra I., Kravchenko, Irina N., Rasskazova, Ekaterina A., Salmova, Margarita A., Tukhovskaya, Elena A., Rykov, Vladimir A., Slashcheva, Gulsara A., Egorova, Natalya S., Muzyka, Inessa S., Tsetlin, Victor I., Utkin, Yuri N.
Formato:	Online Artículo Texto
Lenguaje:	English
Publicado:	MDPI 2018
Materias:	Article
Acceso en línea:	https://www.ncbi.nlm.nih.gov/pmc/articles/PMC5793121/ https://www.ncbi.nlm.nih.gov/pubmed/29316656 http://dx.doi.org/10.3390/toxins10010034

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