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[(18)F]Fluorophenylazocarboxylates: Design and Synthesis of Potential Radioligands for Dopamine D3 and μ-Opioid Receptor

[Image: see text] (18)F-Labeled building blocks from the type of [(18)F]fluorophenylazocarboxylic-tert-butyl esters offer a rapid, mild, and reliable method for the (18)F-fluoroarylation of biomolecules. Two series of azocarboxamides were synthesized as potential radioligands for dopamine D3 and the...

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Detalles Bibliográficos
Autores principales:	Nebel, Natascha, Strauch, Brigitte, Maschauer, Simone, Lasch, Roman, Rampp, Hannelore, Fehler, Stefanie K., Bock, Leonard R., Hübner, Harald, Gmeiner, Peter, Heinrich, Markus R., Prante, Olaf
Formato:	Online Artículo Texto
Lenguaje:	English
Publicado:	American Chemical Society 2017
Acceso en línea:	https://www.ncbi.nlm.nih.gov/pmc/articles/PMC5819854/ https://www.ncbi.nlm.nih.gov/pubmed/29479577 http://dx.doi.org/10.1021/acsomega.7b01374

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