Cargando…

Microwave-assisted synthesis and bioevaluation of new sulfonamides

In this study, 4-[5-(4-hydroxyphenyl)-3-aryl-4,5-dihydro-1H-pyrazol-1-yl]benzenesulfonamide derivatives (8-14) were synthesized for the first time by microwave irradiation and their chemical structures were confirmed by (1)H NMR, (13)C NMR and HRMS. Cytotoxic activities and inhibitory effects on car...

Descripción completa

Detalles Bibliográficos
Autores principales:	Gul, Halise Inci, Yamali, Cem, Yesilyurt, Fatma, Sakagami, Hiroshi, Kucukoglu, Kaan, Gulcin, Ilhami, Gul, Mustafa, Supuran, Claudiu T.
Formato:	Online Artículo Texto
Lenguaje:	English
Publicado:	Taylor & Francis 2017
Materias:	Research Article
Acceso en línea:	https://www.ncbi.nlm.nih.gov/pmc/articles/PMC6009867/ https://www.ncbi.nlm.nih.gov/pubmed/28260401 http://dx.doi.org/10.1080/14756366.2016.1254207

Ejemplares similares

Designing, synthesis and bioactivities of 4-[3-(4-hydroxyphenyl)-5-aryl-4,5-dihydro-pyrazol-1-yl]benzenesulfonamides
por: Gul, Halise Inci, et al.
Publicado: (2016)

Synthesis and bioactivities of 1-(4-hydroxyphenyl)-2-((heteroaryl)thio)ethanones as carbonic anhydrase I, II and acetylcholinesterase inhibitors
por: YAMALI, Cem, et al.
Publicado: (2020)

Synthesis, cytotoxicities, and carbonic anhydrase inhibition potential of 6-(3-aryl-2-propenoyl)-2(3H)-benzoxazolones
por: Bilginer, Sinan, et al.
Publicado: (2019)

Synthesis, carbonic anhydrase I and II inhibition studies of the 1,3,5-trisubstituted-pyrazolines
por: Gul, Halise Inci, et al.
Publicado: (2016)

Synthesis and biological evaluation of new pyrazolebenzene-sulphonamides as potential anticancer agents and hCA I and II inhibitors
por: TUĞRAK, Mehtap, et al.
Publicado: (2021)

Novel sulphonamides incorporating triazene moieties show powerful carbonic anhydrase I and II inhibitory properties
por: Bilginer, Sinan, et al.
Publicado: (2019)

Synthesis and pharmacological effects of novel benzenesulfonamides carrying benzamide moiety as carbonic anhydrase and acetylcholinesterase inhibitors
por: TUĞRAK, Mehtap, et al.
Publicado: (2020)

Crystal structure and theoretical study of (2E)-1-[4-hydroxy-3-(morpholin-4-ylmethyl)phenyl]-3-(thiophen-2-yl)prop-2-en-1-one
por: Yesilyurt, Fatma, et al.
Publicado: (2018)

Special Issue: Sulfonamides
por: Supuran, Claudiu T.
Publicado: (2017)

Natural-Product-Inspired Microwave-Assisted Synthesis of Novel Spirooxindoles as Antileishmanial Agents: Synthesis, Stereochemical Assignment, Bioevaluation, SAR, and Molecular Docking Studies
por: Sahu, Nawal Kishore, et al.
Publicado: (2023)

Synthesis and bioactivity of several new hetaryl sulfonamides
por: Taslimi, Parham, et al.
Publicado: (2017)

Synthesis and cytotoxic activities of novel copper and silver complexes of 1,3-diaryltriazene-substituted sulfonamides
por: Canakci, Dilek, et al.
Publicado: (2018)

Five-Membered Heterocyclic Sulfonamides as Carbonic Anhydrase Inhibitors
por: Angeli, Andrea, et al.
Publicado: (2023)

Secondary Sulfonamides as Effective Lactoperoxidase Inhibitors
por: Köksal, Zeynep, et al.
Publicado: (2017)

Monoamine Oxidase (MAO) as a Potential Target for Anticancer Drug Design and Development
por: Aljanabi, Reem, et al.
Publicado: (2021)

Terminators or Guardians? Design, Synthesis, and Cytotoxicity Profiling of Chalcone-Sulfonamide Hybrids
por: Aboukhatwa, Shaimaa M., et al.
Publicado: (2023)

Synthesis, Preliminary Bioevaluation and Computational Analysis of Caffeic Acid Analogues
por: Liu, Zhiqian, et al.
Publicado: (2014)

Design, Synthesis and in Combo Antidiabetic Bioevaluation of Multitarget Phenylpropanoic Acids †
por: Colín-Lozano, Blanca, et al.
Publicado: (2018)

Synthesis of an acridine orange sulfonamide derivative with potent carbonic anhydrase IX inhibitory action
por: Bragagni, Marco, et al.
Publicado: (2017)

Assessment of the antiproliferative and apoptotic roles of sulfonamide carbonic anhydrase IX inhibitors in HeLa cancer cell line
por: Koyuncu, Ismail, et al.
Publicado: (2018)

3-(4-Chlorobenzoyl)-4-(4-chlorophenyl)-1-phenethylpiperidin-4-ol
por: Aydın, Abdullah, et al.
Publicado: (2011)

N-[2-(4-Bromobenzoyl)ethyl]isopropylaminium chloride
por: Aydın, Abdullah, et al.
Publicado: (2011)

N-(2-Benzoylethyl)propan-2-aminium chloride
por: Aydın, Abdullah, et al.
Publicado: (2012)

N-[2-(4-Methylbenzoyl)ethyl]propan-2-aminium chloride
por: Aydın, Abdullah, et al.
Publicado: (2012)

New sulfonamides containing organometallic-acylhydrazones: synthesis, characterisation and biological evaluation as inhibitors of human carbonic anhydrases
por: Huentupil, Yosselin, et al.
Publicado: (2019)

Synthesis, Bioevaluation and Molecular Dynamic Simulation Studies of Dexibuprofen–Antioxidant Mutual Prodrugs
por: Ashraf, Zaman, et al.
Publicado: (2016)

Synthesis and bioevaluation of novel steroidal isatin conjugates derived from epiandrosterone/androsterone
por: Ke, Shaoyong, et al.
Publicado: (2019)

Design, synthesis and bioevaluation of novel 6-substituted aminoindazole derivatives as anticancer agents
por: Hoang, Ngo Xuan, et al.
Publicado: (2020)

Benzamide-4-Sulfonamides Are Effective Human Carbonic Anhydrase I, II, VII, and IX Inhibitors
por: Abdoli, Morteza, et al.
Publicado: (2018)

The palladium-based complexes bearing 1,3-dibenzylbenzimidazolium with morpholine, triphenylphosphine, and pyridine derivate ligands: synthesis, characterization, structure and enzyme inhibitions
por: Aktaş, Aydın, et al.
Publicado: (2022)

Carbonic Anhydrase Inhibitors. Part 54(1): Metal Complexes of Heterocyclic Sulfonamides: A New Class of Antiglaucoma Agents
por: Supuran, Claudiu T., et al.
Publicado: (1997)

Structural Basis for the Inhibition of Helicobacter pylori α-Carbonic Anhydrase by Sulfonamides
por: Modakh, Joyanta K., et al.
Publicado: (2015)

Discovery of novel 1,3-diaryltriazene sulfonamides as carbonic anhydrase I, II, VII, and IX inhibitors
por: Akocak, Suleyman, et al.
Publicado: (2018)

Synthesis and Antifungal Evaluation of 1-Aryl-2-dimethyl- aminomethyl-2-propen-1-one Hydrochlorides
por: Mete, Ebru, et al.
Publicado: (2011)

DNA-Binding Interaction Studies of Microwave Assisted Synthesized Sulfonamide Substituted 8-Hydroxyquinoline Derivatives
por: Dixit, Ritu B., et al.
Publicado: (2011)

Synthesis and biological evaluation of aminomethyl and alkoxymethyl derivatives as carbonic anhydrase, acetylcholinesterase and butyrylcholinesterase inhibitors
por: Gulçin, İlhami, et al.
Publicado: (2017)

Pyrazolo[4,3-c]pyridine Sulfonamides as Carbonic Anhydrase Inhibitors: Synthesis, Biological and In Silico Studies
por: Angeli, Andrea, et al.
Publicado: (2022)

Synthesis of Sulfonamides Incorporating Piperidinyl-Hydrazidoureido and Piperidinyl-Hydrazidothioureido Moieties and Their Carbonic Anhydrase I, II, IX and XII Inhibitory Activity
por: Moi, Davide, et al.
Publicado: (2022)

Design, synthesis, and bioevaluation of viral 3C and 3C-like protease inhibitors
por: Prior, Allan M., et al.
Publicado: (2013)

Crystal structure of 1-{4-hydroxy-3-[(pyrrolidin-1-yl)methyl]phenyl}-3-phenylprop-2-en-1-one
por: Aydın, Abdullah, et al.
Publicado: (2016)

Cannot write session to /tmp/vufind_sessions/sess_ocoilcapd3n2shdr9viuiiro3h