Convenient Synthesis of Thiohydantoins, Imidazole-2-thiones and Imidazo[2,1-b]thiazol-4-iums from Polymer-Supported α-Acylamino Ketones

The preparation of 5-methylene-thiohydantoins using solid-phase synthesis is reported in this paper. After sulfonylation of immobilized Ser (t-Bu)-OH with 4-nitrobenzenesulfonyl chloride followed by alkylation with various bromoketones, the 4-Nos group was removed and the resulting polymer-supported...

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Detalles Bibliográficos
Autores principales: Králová, Petra, Maloň, Michal, Koshino, Hiroyuki, Soural, Miroslav
Formato: Online Artículo Texto
Lenguaje:English
Publicado: MDPI 2018
Materias:
Article
Acceso en línea:https://www.ncbi.nlm.nih.gov/pmc/articles/PMC6017016/
https://www.ncbi.nlm.nih.gov/pubmed/29690582
http://dx.doi.org/10.3390/molecules23040976

Internet

https://www.ncbi.nlm.nih.gov/pmc/articles/PMC6017016/
https://www.ncbi.nlm.nih.gov/pubmed/29690582
http://dx.doi.org/10.3390/molecules23040976

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