Cargando…

Design, Synthesis and DFT/DNP Modeling Study of New 2-Amino-5-arylazothiazole Derivatives as Potential Antibacterial Agents

A new series of 2-amino-5-arylazothiazole derivatives has been designed and synthesized in 61–78% yields and screened as potential antibacterial drug candidates against the Gram negative bacterium Escherichia coli. The geometry of the title compounds were being studied using the Material Studio pack...

Descripción completa

Detalles Bibliográficos
Autor principal:	Abu-Melha, Sraa
Formato:	Online Artículo Texto
Lenguaje:	English
Publicado:	MDPI 2018
Materias:	Article
Acceso en línea:	https://www.ncbi.nlm.nih.gov/pmc/articles/PMC6017174/ https://www.ncbi.nlm.nih.gov/pubmed/29462895 http://dx.doi.org/10.3390/molecules23020434

Ejemplares similares

Pyridyl thiosemicarbazide: synthesis, crystal structure, DFT/B3LYP, molecular docking studies and its biological investigations
por: Abu-Melha, Sraa
Publicado: (2018)

Synthesis of Some Novel 2-Amino-5-arylazothiazole Disperse Dyes for Dyeing Polyester Fabrics and Their Antimicrobial Activity
por: Gaffer, Hatem E., et al.
Publicado: (2016)

Eco-Friendly Synthesis of Some Thiosemicarbazones and Their Applications as Intermediates for 5-Arylazothiazole Disperse Dyes
por: Gaffer, Hatem E., et al.
Publicado: (2015)

Synthesis and Biological Evaluation of Some Novel Thiazole-Based Heterocycles as Potential Anticancer and Antimicrobial Agents
por: Abu-Melha, Sraa, et al.
Publicado: (2019)

Eco-Friendly Synthesis, Characterization and Biological Evaluation of Some Novel Pyrazolines Containing Thiazole Moiety as Potential Anticancer and Antimicrobial Agents
por: Edrees, Mastoura M., et al.
Publicado: (2018)

Dendritic polarizing agents for DNP SENS
por: Liao, Wei-Chih, et al.
Publicado: (2017)

Potential COVID-19 Drug Candidates Based on Diazinyl-Thiazol-Imine Moieties: Synthesis and Greener Pastures Biological Study
por: Abu-Melha, Sraa, et al.
Publicado: (2022)

Synthesis and Antimicrobial Activity of Some New Thiadiazoles, Thioamides, 5-Arylazothiazoles and Pyrimido[4,5-d][1,2,4]triazolo[4,3-a]pyrimidines
por: Abdelhamid, Abdou O., et al.
Publicado: (2016)

DNP 2017
Publicado: (2017)

Design, Synthesis and Evaluation of the Antibacterial Enhancement Activities of Amino Dihydroartemisinin Derivatives
por: Wu, Chong, et al.
Publicado: (2013)

An Enhanced Actualized DNP Model to Improve DNP Project Placements, Rigor, and Completion
por: VanderKooi, Marie E., et al.
Publicado: (2018)

Design, Modeling and Synthesis of 1,2,3-Triazole-Linked Nucleoside-Amino Acid Conjugates as Potential Antibacterial Agents
por: Malkowski, Sarah N., et al.
Publicado: (2017)

Clean Grinding Technique: A Facile Synthesis and In Silico Antiviral Activity of Hydrazones, Pyrazoles, and Pyrazines Bearing Thiazole Moiety against SARS-CoV-2 Main Protease (M(pro))
por: Abu-Melha, Sraa, et al.
Publicado: (2020)

Leadership and systems improvement for the DNP
por: Armstrong, Gail, et al.
Publicado: (2019)

Design, Synthesis, DFT Study and Antifungal Activity of Pyrazolecarboxamide Derivatives
por: Mu, Jin-Xia, et al.
Publicado: (2016)

A facile sonochemical protocol for synthesis of 3-amino- and 4-amino-1,2,4-triazole derived Schiff bases as potential antibacterial agents
por: Sultan, Aeysha, et al.
Publicado: (2020)

Monomyristin and Monopalmitin Derivatives: Synthesis and Evaluation as Potential Antibacterial and Antifungal Agents
por: Jumina,, et al.
Publicado: (2018)

Design, Synthesis, Molecular Docking, and Antibacterial Evaluation of Some Novel Flouroquinolone Derivatives as Potent Antibacterial Agent
por: Patel, Mehul M., et al.
Publicado: (2014)

Design, Synthesis and Biological Evaluation of Lophanic Acid Derivatives as Antifungal and Antibacterial Agents
por: Yu, Xiang, et al.
Publicado: (2022)

Influence of DNP Polarizing Agents on Biochemical Processes: TEMPOL in Transient Ischemic Stroke
por: Lê, Thanh Phong, et al.
Publicado: (2023)

Discovery of Quinazoline-2,4(1H,3H)-Dione Derivatives as Potential Antibacterial Agent: Design, Synthesis, and Their Antibacterial Activity
por: Boshta, Nader M., et al.
Publicado: (2022)

Continuous-flow DNP polarizer for MRI applications at 1.5 T
por: Denysenkov, V., et al.
Publicado: (2017)

Retraction: A facile sonochemical protocol for synthesis of 3-amino- and 4-amino-1,2,4-triazole derived Schiff bases as potential antibacterial agents
Publicado: (2020)

Synthesis and Antimicrobial Evaluation of 1,4‐Naphthoquinone Derivatives as Potential Antibacterial Agents
por: Ravichandiran, Palanisamy, et al.
Publicado: (2019)

DNp73: oncotarget in invasion and metastasis
por: Pützer, Brigitte M.
Publicado: (2013)

Design, Synthesis, and Structure–Activity Relationship Studies of New Quinone Derivatives as Antibacterial Agents
por: Andrades-Lagos, Juan, et al.
Publicado: (2023)

STUDIES ON ARTIFICIAL ANTIGENS : I. ANTIGENICITY OF DNP-POLYLYSINE AND DNP COPOLYMER OF LYSINE AND GLUTAMIC ACID IN GUINEA PIGS
por: Kantor, Fred S., et al.
Publicado: (1963)

Synthesis, DFT investigations, antioxidant, antibacterial activity and SAR-study of novel thiophene-2-carboxamide derivatives
por: Metwally, Heba M., et al.
Publicado: (2023)

Novel Quinoline-Based Thiosemicarbazide Derivatives: Synthesis, DFT Calculations, and Investigation of Antitubercular, Antibacterial, and Antifungal Activities
por: Özcan, Esma, et al.
Publicado: (2023)

Synthesis and Biological Evaluation of Fingolimod Derivatives as Antibacterial Agents
por: Zore, Matej, et al.
Publicado: (2021)

Design, Synthesis, and Evaluation of Amphiphilic Cyclic and Linear Peptides Composed of Hydrophobic and Positively-Charged Amino Acids as Antibacterial Agents
por: Riahifard, Neda, et al.
Publicado: (2018)

Towards Anticancer and Antibacterial Agents: Design and Synthesis of 1,2,3-Triazol-quinobenzothiazine Derivatives
por: Kisiel-Nawrot, Ewa, et al.
Publicado: (2023)

Jacqueline Herd DNP, RN, NEA-BC
por: Shinkus Clark, Joan
Publicado: (2020)

Targeted DNP for biomolecular solid-state NMR
por: Gauto, Diego, et al.
Publicado: (2021)

A STUDY OF THE PASSIVE TRANSFER OF DELAYED HYPERSENSITIVITY TO DNP-POLY-L-LYSINE AND DNP-GL IN RESPONDER AND NONRESPONDER GUINEA PIGS
por: Green, Ira, et al.
Publicado: (1967)

Quenching of Tryptophan Fluorescence in the Presence of 2,4-DNP, 2,6-DNP, 2,4-DNA and DNOC and Their Mechanism of Toxicity
por: Huţanu, Cristina-Amalia Dumitraş, et al.
Publicado: (2013)

Practical modern SCADA protocols: DNP3, 60870.5 and related systems
por: Clarke, Gordon R, et al.
Publicado: (2004)

Design, Synthesis of Novel Tetrandrine-14-l-Amino Acid and Tetrandrine-14-l-Amino Acid-Urea Derivatives as Potential Anti-Cancer Agents
por: Hu, Sheng-Cao, et al.
Publicado: (2020)

Design, synthesis and antiproliferative screening of newly synthesized acrylate derivatives as potential anticancer agents
por: Alshaya, Dalal Sulaiman, et al.
Publicado: (2023)

Design and Synthesis of Benzimidazole-Chalcone Derivatives as Potential Anticancer Agents
por: Hsieh, Cheng-Ying, et al.
Publicado: (2019)

Cannot write session to /tmp/vufind_sessions/sess_j8mal8vg3ahtofu98nuhia6omn