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First Metal-Free Synthesis of Tetracyclic Pyrido and Pyrazino Thienopyrimidinone Molecules

We report herein a new metal free synthetic pathway to generate tetracyclic compounds from 3-aminothieno[3,2-b]pyridine-2-carboxylate. To enlarge the molecular diversity, we studied the Suzuki coupling of 9-chloro-6H-pyrido[1,2-a]pyrido[2′,3′:4,5]thieno[3,2-d]pyrimidin-6-one and several boronic acid...

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Detalles Bibliográficos
Autores principales:	Aounzou, Mohammed, Campos, Joana F., Loubidi, Mohammed, Berteina-Raboin, Sabine
Formato:	Online Artículo Texto
Lenguaje:	English
Publicado:	MDPI 2018
Materias:	Article
Acceso en línea:	https://www.ncbi.nlm.nih.gov/pmc/articles/PMC6100531/ https://www.ncbi.nlm.nih.gov/pubmed/29751677 http://dx.doi.org/10.3390/molecules23051159

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