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Short and Efficient Synthesis of Optically Active N-Tosyl Aziridines from 2-Amino Alcohols
Two alternative and complementary one-pot procedures for the direct transformation of 2-amino alcohols to N-tosyl aziridines are presented. The unsubstituted parent compound and its less hindered homologues can be obtained in high yields by tosylation and in situ cyclisation effected by potassium hy...
Autores principales: | Bieber, Lothar W., de Araújo, Maria C. F. |
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Formato: | Online Artículo Texto |
Lenguaje: | English |
Publicado: |
MDPI
2002
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Materias: | |
Acceso en línea: | https://www.ncbi.nlm.nih.gov/pmc/articles/PMC6146485/ http://dx.doi.org/10.3390/71200902 |
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