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New Bioactive Azaartemisinin Derivatives

Reaction of artemisinin (1) with ethanolamine, followed by acid treatment produced the lactam (4S,8S,9S,13S,1R,5R,12R)-11-aza-11-(2-hydroxyethyl)-1,5,9-trimethyl-14,15-dioxatetracyclo [10.2.1.0<4,13>.0<8,13>]pentadecan-10-one (4) and the diol (1S,2S,6S,7S,5R,8R)-4-aza-5,6-dihydroxy-4-(2-...

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Detalles Bibliográficos
Autores principales:	Al-Oqail, Mai M., Galal, Ahmed M., Ahmad, Mohamed S., Al-Fishawi, Ahlam M., El-Feraly, Farouk S.
Formato:	Online Artículo Texto
Lenguaje:	English
Publicado:	MDPI 2003
Materias:	Article
Acceso en línea:	https://www.ncbi.nlm.nih.gov/pmc/articles/PMC6146936/ http://dx.doi.org/10.3390/81200901

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