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An Affinity-Based Probe for the Human Adenosine A(2A) Receptor

[Image: see text] Using activity-based protein profiling (ABPP), functional proteins can be interrogated in their native environment. Despite their pharmaceutical relevance, G protein-coupled receptors (GPCRs) have been difficult to address through ABPP. In the current study, we took the prototypica...

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Detalles Bibliográficos
Autores principales:	Yang, Xue, Michiels, Thomas J. M., de Jong, Coen, Soethoudt, Marjolein, Dekker, Niek, Gordon, Euan, van der Stelt, Mario, Heitman, Laura H., van der Es, Daan, IJzerman, Adriaan P.
Formato:	Online Artículo Texto
Lenguaje:	English
Publicado:	American Chemical Society 2018
Acceso en línea:	https://www.ncbi.nlm.nih.gov/pmc/articles/PMC6150691/ https://www.ncbi.nlm.nih.gov/pubmed/30080404 http://dx.doi.org/10.1021/acs.jmedchem.8b00860

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