Cargando…
Chloroquine analogs as antimalarial candidates with potent in vitro and in vivo activity
In spite of recent efforts to eradicate malaria in the world, this parasitic disease is still considered a major public health problem, with a total of 216 million cases of malaria and 445,000 deaths in 2016. Artemisinin-based combination therapies remain effective in most parts of the world, but re...
Autores principales: | Aguiar, Anna C.C., Murce, Erika, Cortopassi, Wilian A., Pimentel, Andre S., Almeida, Maria M.F.S., Barros, Daniele C.S., Guedes, Jéssica S., Meneghetti, Mario R., Krettli, Antoniana U. |
---|---|
Formato: | Online Artículo Texto |
Lenguaje: | English |
Publicado: |
Elsevier
2018
|
Materias: | |
Acceso en línea: | https://www.ncbi.nlm.nih.gov/pmc/articles/PMC6215995/ https://www.ncbi.nlm.nih.gov/pubmed/30396013 http://dx.doi.org/10.1016/j.ijpddr.2018.10.002 |
Ejemplares similares
-
Antimalarial Activity and Mechanisms of Action of Two Novel 4-Aminoquinolines against Chloroquine-Resistant Parasites
por: Aguiar, Anna Caroline Campos, et al.
Publicado: (2012) -
Fighting Plasmodium chloroquine resistance with acetylenic chloroquine analogues
por: Cortopassi, Wilian A., et al.
Publicado: (2022) -
Antimalarial Activity of Potential Inhibitors of Plasmodium falciparum Lactate Dehydrogenase Enzyme Selected by Docking Studies
por: Penna-Coutinho, Julia, et al.
Publicado: (2011) -
Antiplasmodial activity of chloroquine analogs against chloroquine-resistant parasites, docking studies and mechanisms of drug action
por: de Souza, Nicolli B, et al.
Publicado: (2014) -
Commercial drugs containing flavonoids are active in mice with
malaria and in vitro against chloroquine-resistant
Plasmodium falciparum
por: Penna-Coutinho, Julia, et al.
Publicado: (2018)