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FSCPX, a Chemical Widely Used as an Irreversible A(1) Adenosine Receptor Antagonist, Modifies the Effect of NBTI, a Nucleoside Transport Inhibitor, by Reducing the Interstitial Adenosine Level in the Guinea Pig Atrium
Based on in silico results, recently we have assumed that FSCPX, an irreversible A(1) adenosine receptor antagonist, inhibits the action of NBTI that is apparent on E/c curves of adenosine receptor agonists. As a mechanism for this unexpected effect, we hypothesized that FSCPX might modify the equil...
Autores principales: | Erdei, Tamas, Szabo, Adrienn Monika, Lampe, Nora, Szabo, Katalin, Kiss, Rita, Zsuga, Judit, Papp, Csaba, Pinter, Akos, Szentmiklosi, Andras Jozsef, Szilvassy, Zoltan, Juhasz, Bela, Gesztelyi, Rudolf |
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Formato: | Online Artículo Texto |
Lenguaje: | English |
Publicado: |
MDPI
2018
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Materias: | |
Acceso en línea: | https://www.ncbi.nlm.nih.gov/pmc/articles/PMC6225130/ https://www.ncbi.nlm.nih.gov/pubmed/30200192 http://dx.doi.org/10.3390/molecules23092186 |
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