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2-Amino- and 2-Alkylthio-4H-3,1-benzothiazin-4-ones: Synthesis, Interconversion and Enzyme Inhibitory Activities

The synthetic access to 2-sec-amino-4H-3,1-benzothiazin-4-ones 2 was explored. Compounds 2 were available from methyl 2-thioureidobenzoates 1, 2-thioureidobenzoic acids 3, and novel 2-thioureidobenzamides 6, respectively, under different conditions. 2-Alkylthio-4H-3,1-benzothiazin-4-ones 5 have been...

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Detalles Bibliográficos
Autores principales:	Häcker, Hans-Georg, Grundmann, Florian, Lohr, Friederike, Ottersbach, Philipp A., Zhou, Jing, Schnakenburg, Gregor, Gütschow, Michael
Formato:	Online Artículo Texto
Lenguaje:	English
Publicado:	Molecular Diversity Preservation International 2009
Materias:	Article
Acceso en línea:	https://www.ncbi.nlm.nih.gov/pmc/articles/PMC6253953/ https://www.ncbi.nlm.nih.gov/pubmed/19145216 http://dx.doi.org/10.3390/molecules14010378

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