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Carnitine Conjugate of Nipecotic Acid: A New Example of Dual Prodrug
As a novel example of improved entry of poorly delivered drugs into the brain by means of nutrient conjugates, L-carnitine was conjugated to nipecotic acid and the capacity to antagonize PTZ-induced convulsions of this novel entity was evaluated.
Autores principales: | Napolitano, Carmela, Scaglianti, Martina, Scalambra, Emanuela, Manfredini, Stefano, Ferraro, Luca, Beggiato, Sarah, Vertuani, Silvia |
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Formato: | Online Artículo Texto |
Lenguaje: | English |
Publicado: |
Molecular Diversity Preservation International
2009
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Materias: | |
Acceso en línea: | https://www.ncbi.nlm.nih.gov/pmc/articles/PMC6255320/ https://www.ncbi.nlm.nih.gov/pubmed/19783924 http://dx.doi.org/10.3390/molecules14093268 |
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