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Synthesis of Novel Aryl(heteroaryl)sulfonyl Ureas of Possible Biological Interest

The course of reaction of aryl and heteroaryl sulfonamides with diphenylcarbonate (DPC) and 4-dimethylaminopyridine (DMAP) was found to depend on the pKa of the sulfonamide used. Aryl sulfonamides with pK(a) ~ 10 gave 4-dimethylamino-pyridinium arylsulfonyl-carbamoylides, while the more acidic heter...

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Detalles Bibliográficos
Autores principales:	Sączewski, Franciszek, Kuchnio, Anna, Samsel, Monika, Łobocka, Marta, Kiedrowska, Agnieszka, Lisewska, Karolina, Sączewski, Jarosław, Gdaniec, Maria, Bednarski, Patrick J.
Formato:	Online Artículo Texto
Lenguaje:	English
Publicado:	Molecular Diversity Preservation International 2010
Materias:	Article
Acceso en línea:	https://www.ncbi.nlm.nih.gov/pmc/articles/PMC6257353/ https://www.ncbi.nlm.nih.gov/pubmed/20335967 http://dx.doi.org/10.3390/molecules15031113

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