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Synthesis and Biological Evaluation of Pyrazolo[1,5-a]-pyrimidine-containing (99m)Tc Nitrido Radiopharmaceuticals as Imaging Agents for Tumors

The compound 5-((2-aminoethylamino)methyl)-7-(4-bromoanilino)-3-cyano-pyrazolo[1,5-a]pyrimidine (ABCPP) was synthesized and conjugated with N-mercapto-acetylglycine (MAG), N-mercaptoacetylphenylalanine (MAF) and N-mercaptoacetylvaline (MAA), respectively. These three compounds were labeled successfu...

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Detalles Bibliográficos
Autores principales:	Ding, Rui, He, Yong, Xu, Jingli, Liu, Hang, Wang, Xiao, Feng, Man, Qi, Chuanmin, Zhang, Junbo
Formato:	Online Artículo Texto
Lenguaje:	English
Publicado:	MDPI 2010
Materias:	Article
Acceso en línea:	https://www.ncbi.nlm.nih.gov/pmc/articles/PMC6259132/ https://www.ncbi.nlm.nih.gov/pubmed/21119567 http://dx.doi.org/10.3390/molecules15128723

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