Cargando…

Synthesis and in Vitro Antimicrobial Activity of Some Pyrazolyl-1-carboxamide Derivatives

A series of 3,5-disubstituted pyrazole-1-carboxamides were obtained by treatment of chalcones with semicarbazide hydrochloride in dioxane containing sodium acetate/acetic acid as a buffer solution. N-acetyl derivatives of pyrazole-1-carboxamides were isolated in good yields either by treatment of th...

Descripción completa

Detalles Bibliográficos
Autores principales:	Sharshira, Essam Mohamed, Hamada, Nagwa Mohamed Mahrous
Formato:	Online Artículo Texto
Lenguaje:	English
Publicado:	MDPI 2011
Materias:	Article
Acceso en línea:	https://www.ncbi.nlm.nih.gov/pmc/articles/PMC6264426/ https://www.ncbi.nlm.nih.gov/pubmed/21909057 http://dx.doi.org/10.3390/molecules16097736

Ejemplares similares

Synthesis and Antimicrobial Evaluation of Some Pyrazole Derivatives
por: Sharshira, Essam Mohamed, et al.
Publicado: (2012)

Synthesis and Antimicrobial Evaluation of Some Heterocyclic Chalcone Derivatives
por: Hamada, Nagwa Mohamed Mahrous, et al.
Publicado: (2011)

Synthesis of Oxadiazolyl, Pyrazolyl and Thiazolyl Derivatives of Thiophene-2-Carboxamide as Antimicrobial and Anti-HCV Agents
por: Rizk, Ola H., et al.
Publicado: (2017)

Synthesis, Characterization, Antimicrobial Screening and Free-Radical Scavenging Activity of Some Novel Substituted Pyrazoles
por: Hamada, Nagwa Mohamed Mahrous, et al.
Publicado: (2015)

Synthesis of Some New Pyridine-2,6-carboxamide-derived Schiff Bases as Potential Antimicrobial Agents
por: Al-Omar, Mohamed A., et al.
Publicado: (2010)

Design, Synthesis, and Antimicrobial Evaluation of Novel Pyrazoles and Pyrazolyl 1,3,4-Thiadiazine Derivatives
por: Radini, Ibrahim Ali M.
Publicado: (2018)

Derivatives of 3-Aminopyrazine-2-carboxamides: Synthesis, Antimicrobial Evaluation, and in Vitro Cytotoxicity
por: Bouz, Ghada, et al.
Publicado: (2019)

Synthesis and Anti-Breast Cancer Potency of Mono- and Bis-(pyrazolyl[1,2,4]triazolo[3,4-b][1,3,4]thiadiazine) Derivatives as EGFR/CDK-2 Target Inhibitors
por: Salem, Mostafa E., et al.
Publicado: (2023)

Synthesis and Biological Evaluation of N- Pyrazolyl Derivatives and Pyrazolopyrimidine Bearing a Biologically Active Sulfonamide Moiety as Potential Antimicrobial Agent
por: Hafez, Hend N., et al.
Publicado: (2016)

Multistep Synthesis and In Vitro Anticancer Evaluation of 2-Pyrazolyl-Estradiol Derivatives, Pyrazolocoumarin-Estradiol Hybrids and Analogous Compounds
por: Molnár, Barnabás, et al.
Publicado: (2020)

Synthesis, Structural Elucidation, and In Vitro Antitumor Activities of Some Pyrazolopyrimidines and Schiff Bases Derived from 5-Amino-3-(arylamino)-1H-pyrazole-4-carboxamides
por: Hafez, Taghrid S., et al.
Publicado: (2013)

Challenging inflammatory process at molecular, cellular and in vivo levels via some new pyrazolyl thiazolones
por: Elzahhar, Perihan A., et al.
Publicado: (2021)

Biological evaluation of pyrazolyl-urea and dihydro-imidazo-pyrazolyl-urea derivatives as potential anti-angiogenetic agents in the treatment of neuroblastoma
por: Marengo, Barbara, et al.
Publicado: (2020)

Synthesis and Antimicrobial Activity of Some New 1,3,4-Thiadiazole Derivatives
por: Farghaly, Thoraya A., et al.
Publicado: (2012)

Synthesis, characterization and pharmacological evaluation of pyrazolyl urea derivatives as potential anti-inflammatory agents
por: Somakala, Kanagasabai, et al.
Publicado: (2017)

Novel Novolac Phenolic Polymeric Network of Chalcones: Synthesis, Characterization, and Thermal–Electrical Conductivity Investigation
por: Sharshira, Essam Mohamed, et al.
Publicado: (2022)

Correction: Biological evaluation of pyrazolyl-urea and dihydro-imidazo-pyrazolyl-urea derivatives as potential anti-angiogenetic agents in the treatment of neuroblastoma
por: Marengo, Barbara, et al.
Publicado: (2023)

Synthesis and Characterization of Some New Bis-Pyrazolyl-Thiazoles Incorporating the Thiophene Moiety as Potent Anti-Tumor Agents
por: Gomha, Sobhi M., et al.
Publicado: (2016)

Microwave Assisted Synthesis of Some New Heterocyclic Spiro-Derivatives with Potential Antimicrobial and Antioxidant Activity
por: Youssef, Mohamed Mohamed, et al.
Publicado: (2010)

Synthesis of Novel Pyrazinamide Derivatives Based on 3-Chloropyrazine-2-carboxamide and Their Antimicrobial Evaluation
por: Jandourek, Ondrej, et al.
Publicado: (2017)

Synthesis of new pyrazolyl-2, 4-thiazolidinediones as antibacterial and antifungal agents
por: Aneja, Deepak K, et al.
Publicado: (2011)

Synthesis and Biological Activity Evaluation of Coumarin-3-Carboxamide Derivatives
por: Phutdhawong, Weerachai, et al.
Publicado: (2021)

Design, Synthesis and Bioactivities of Novel 1,4-Pentadien-3-one Derivatives Containing a Substituted Pyrazolyl Moiety
por: Chen, Cuili, et al.
Publicado: (2017)

Fe(III) Complexes Based on Mono- and Bis-pyrazolyl-s-triazine Ligands: Synthesis, Molecular Structure, Hirshfeld, and Antimicrobial Evaluations
por: Soliman, Saied M., et al.
Publicado: (2020)

New Thiophenyl-pyrazolyl-thiazole Hybrids as DHFR Inhibitors: Design, Synthesis, Antimicrobial Evaluation, Molecular Modeling, and Biodistribution Studies
por: Dawood, Dina H., et al.
Publicado: (2023)

Synthesis and Antimicrobial Activity of a New Series of Thiazolidine-2,4-diones Carboxamide and Amino Acid Derivatives
por: Abd Alhameed, Rakia, et al.
Publicado: (2019)

Diastereoselective synthesis of atropisomeric pyrazolyl pyrrolo[3,4-d]isoxazolidines via pyrazolyl nitrone cycloaddition to facially divergent maleimides: intensive NMR and DFT studies
por: Said, Awad I., et al.
Publicado: (2020)

Synthesis, DFT investigations, antioxidant, antibacterial activity and SAR-study of novel thiophene-2-carboxamide derivatives
por: Metwally, Heba M., et al.
Publicado: (2023)

Synthesis, In Vitro Antimicrobial and Cytotoxic Activities of Some New Pyrazolo[1,5-a]pyrimidine Derivatives
por: Fouda, Ahmed M., et al.
Publicado: (2019)

Synthesis of New Bitopic Tetra(pyrazolyl)-Ligands with Neopentane and O-Xylene Backbones
por: Potapov, Andrei S., et al.
Publicado: (2012)

Synthesis of Known and Previously Inaccessible Poly(pyrazolyl)Borates under Mild Conditions
por: Melero, María M., et al.
Publicado: (2023)

Synthesis and Antimicrobial Activity of Some New Quinoxaline Derivatives
por: Singh, Dharmchand Prasad, et al.
Publicado: (2010)

Synthesis and antimicrobial activity of some new diphenylamine derivatives
por: Kumar, Arvind, et al.
Publicado: (2015)

Synthesis and Antimicrobial Activity of Some Novel Cross-Linked Chitosan Hydrogels
por: Mohamed, Nadia Ahmed, et al.
Publicado: (2012)

Synthesis and Anticonvulsant Activity of Some Quinazolin-4-(3H)-one Derivatives
por: Georgey, Hanan, et al.
Publicado: (2008)

Synthesis of Some Novel Heterocyclic and Schiff Base Derivatives as Antimicrobial Agents
por: Azab, Mohamed E., et al.
Publicado: (2015)

The Pyrazolyl-Urea Gege3 Inhibits the Activity of ANXA1 in the Angiogenesis Induced by the Pancreatic Cancer Derived EVs
por: Belvedere, Raffaella, et al.
Publicado: (2021)

Synthesis and Antimicrobial Activity of Some New Substituted Quinoxalines
por: El-Atawy, Mohamed A., et al.
Publicado: (2019)

Synthesis and anti-nociceptive potential of isoxazole carboxamide derivatives
por: Bibi, Hajira, et al.
Publicado: (2019)

Targeting USP-7 by a Novel Fluorinated 5-Pyrazolyl-Urea Derivative
por: Morretta, Elva, et al.
Publicado: (2023)

Cannot write session to /tmp/vufind_sessions/sess_93o9p987v9i6lfvau9s58chvc9