Cargando…

Synthesis and Antibacterial Activity of Some Heterocyclic Chalcone Analogues Alone and in Combination with Antibiotics

A series of simple heterocyclic chalcone analogues have been synthesized by Claisen Schmidt condensation reactions between substituted benzaldehydes and heteroaryl methyl ketones and evaluated for their antibacterial activity. The structures of the synthesized chalcones were established by IR and (1...

Descripción completa

Detalles Bibliográficos
Autores principales:	Tran, Thanh-Dao, Nguyen, Thi-Thao-Nhu, Do, Tuong-Ha, Huynh, Thi-Ngoc-Phuong, Tran, Cat-Dong, Thai, Khac-Minh
Formato:	Online Artículo Texto
Lenguaje:	English
Publicado:	MDPI 2012
Materias:	Article
Acceso en línea:	https://www.ncbi.nlm.nih.gov/pmc/articles/PMC6268422/ https://www.ncbi.nlm.nih.gov/pubmed/22728362 http://dx.doi.org/10.3390/molecules17066684

Ejemplares similares

Synthesis and Selective Cytotoxic Activities on Rhabdomyosarcoma and Noncancerous Cells of Some Heterocyclic Chalcones
por: Do, Tuong-Ha, et al.
Publicado: (2016)

QSAR Modeling on Benzo[c]phenanthridine Analogues as Topoisomerase I Inhibitors and Anti-cancer Agents
por: Thai, Khac-Minh, et al.
Publicado: (2012)

A Support Vector Machine Classification Model for Benzo[c]phenathridine Analogues with Topoisomerase-I Inhibitory Activity
por: Thai, Khac-Minh, et al.
Publicado: (2012)

Synthesis, In Silico and In Vitro Evaluation for Acetylcholinesterase and BACE-1 Inhibitory Activity of Some N-Substituted-4-Phenothiazine-Chalcones
por: Tran, Thai-Son, et al.
Publicado: (2020)

Exploration of chalcones as 3-chymotrypsin-like protease (3CL(pro)) inhibitors of SARS-CoV-2 using computational approaches
por: Lam, Thua-Phong, et al.
Publicado: (2022)

Chalcone Derivatives as Potential Inhibitors of P-Glycoprotein and NorA: An In Silico and In Vitro Study
por: Le, Minh-Tri, et al.
Publicado: (2022)

Structural Correlation of Some Heterocyclic Chalcone Analogues and Evaluation of Their Antioxidant Potential
por: Kumar, C. S. Chidan, et al.
Publicado: (2013)

Synthesis, In Silico and In Vitro Evaluation of Some Flavone Derivatives for Acetylcholinesterase and BACE-1 Inhibitory Activity
por: Tran, Thai-Son, et al.
Publicado: (2020)

The Effects of One-Point Mutation on the New Delhi Metallo Beta-Lactamase-1 Resistance toward Carbapenem Antibiotics and β-Lactamase Inhibitors: An In Silico Systematic Approach
por: Tran, Van-Thanh, et al.
Publicado: (2022)

Discovery of small molecular inhibitors for interleukin-33/ST2 protein–protein interaction: a virtual screening, molecular dynamics simulations and binding free energy calculations
por: Mai, Tan Thanh, et al.
Publicado: (2022)

A Review of the In Vitro Inhibition of α-Amylase and α-Glucosidase by Chalcone Derivatives
por: Tran, Thanh-Dao, et al.
Publicado: (2023)

Synthesis and Regioselective Reaction of Some Unsymmetrical Heterocyclic Chalcone Derivatives and Spiro Heterocyclic Compounds as Antibacterial Agents
por: El-Hashash, Maher A., et al.
Publicado: (2015)

Identification of small molecules as potential inhibitors of interleukin 6: a multi-computational investigation
por: Tran, Que-Huong, et al.
Publicado: (2022)

Rapid response to the COVID-19 pandemic: Vietnam government’s experience and preliminary success
por: Tran, Thi Phuong Thao, et al.
Publicado: (2020)

Design of Curcumin and Flavonoid Derivatives with Acetylcholinesterase and Beta-Secretase Inhibitory Activities Using in Silico Approaches
por: Tran, Thai-Son, et al.
Publicado: (2020)

Structure-Based Discovery of ABCG2 Inhibitors: A Homology Protein-Based Pharmacophore Modeling and Molecular Docking Approach
por: Le, Minh-Tri, et al.
Publicado: (2021)

Some chalcones derived from thiophene-3-carbaldehyde: synthesis and crystal structures
por: Vu Quoc, Trung, et al.
Publicado: (2019)

Structure-based 3D-Pharmacophore modeling to discover novel interleukin 6 inhibitors: An in silico screening, molecular dynamics simulations and binding free energy calculations
por: Tran, Que-Huong, et al.
Publicado: (2022)

Correction: An efficient multicomponent synthesis of 2,4,5-trisubstituted and 1,2,4,5-tetrasubstituted imidazoles catalyzed by a magnetic nanoparticle supported Lewis acidic deep eutectic solvent
por: Nguyen, Thanh Thi, et al.
Publicado: (2020)

An efficient multicomponent synthesis of 2,4,5-trisubstituted and 1,2,4,5-tetrasubstituted imidazoles catalyzed by a magnetic nanoparticle supported Lewis acidic deep eutectic solvent
por: Nguyen, Thanh Thi, et al.
Publicado: (2019)

Characterizations and Antibacterial Efficacy of Chitosan Oligomers Synthesized by Microwave-Assisted Hydrogen Peroxide Oxidative Depolymerization Method for Infectious Wound Applications
por: Doan, Vinh Khanh, et al.
Publicado: (2021)

Identification of Diosmin and Flavin Adenine Dinucleotide as Repurposing Treatments for Monkeypox Virus: A Computational Study
por: Lam, Thua-Phong, et al.
Publicado: (2022)

Exploring the Mechanism of Subjective Social Status on Compulsive Shopping Behavior: A Moderated Mediation Model of Self-compassion and Depression
por: Tran, Thao Phuong Thi, et al.
Publicado: (2023)

Synthesis and Antimicrobial Evaluation of Some Heterocyclic Chalcone Derivatives
por: Hamada, Nagwa Mohamed Mahrous, et al.
Publicado: (2011)

Optimization of Oligomer Chitosan/Polyvinylpyrrolidone Coating for Enhancing Antibacterial, Hemostatic Effects and Biocompatibility of Nanofibrous Wound Dressing
por: Doan, Vinh Khanh, et al.
Publicado: (2022)

Soy Lecithin-Derived Liposomal Delivery Systems: Surface Modification and Current Applications
por: Le, Ngoc Thuy Trang, et al.
Publicado: (2019)

Reactive Hemophagocytic Lymphohistiocytosis-Associated Kikuchi-Fujimoto Disease After a Staphylococcus epidermidis Cutaneous Infection: The First Case Report
por: Cao, Ngoc Thanh, et al.
Publicado: (2021)

Development of a Cell Suspension Culture System for Promoting Alkaloid and Vinca Alkaloid Biosynthesis Using Endophytic Fungi Isolated from Local Catharanthus roseus
por: Linh, Tran My, et al.
Publicado: (2021)

Heterocyclic amines detected in cooked meats and fishes from street markets and restaurants in the city of Hanoi, Vietnam: A Pilot local field investigation findings in 2020
por: Hao, Le Thi Hong, et al.
Publicado: (2022)

Toxicity Assessments of Chalcone and Some Synthetic Chalcone Analogues in a Zebrafish Model
por: Lee, Ya-Ting, et al.
Publicado: (2014)

Genomic alterations involved in fluoroquinolone resistance development in Staphylococcus aureus
por: Huynh, Thuc Quyen, et al.
Publicado: (2023)

Age distribution of dengue cases in southern Vietnam from 2000 to 2015
por: Taurel, Anne-Frieda, et al.
Publicado: (2023)

Gelatin-stabilized composites of silver nanoparticles and curcumin: characterization, antibacterial and antioxidant study
por: Loan Khanh, Ly, et al.
Publicado: (2019)

Synthesis and characterization of some novel polythiophene derivatives containing pyrazoline
por: Trung, Vu Quoc, et al.
Publicado: (2022)

Application of Essential Oils Extracted from Peel Wastes of Four Orange Varieties to Control Anthracnose Caused by Colletotrichum scovillei and Colletotrichum gloeosporioides on Mangoes
por: Duong, Chau Trung, et al.
Publicado: (2023)

Identification of potential interleukin-8 inhibitors acting on the interactive site between chemokine and CXCR2 receptor: A computational approach
por: Tran, Thi-Thuy-Nga, et al.
Publicado: (2022)

Association between perceived harm of tobacco and intention to quit: a cross-sectional analysis of the Vietnam Global Adult Tobacco Survey
por: Tran, Thi Phuong Thao, et al.
Publicado: (2022)

Mapping for Engagement: Setting up a Community Based Participatory Research Project to Reach Underserved Communities at Risk for Hepatitis C in Ho Chi Minh City, Vietnam
por: Nguyen Quoc, Giang, et al.
Publicado: (2022)

Detection of maternal carriers of common α-thalassemia deletions from cell-free DNA
por: Doan, Phuoc-Loc, et al.
Publicado: (2022)

Age-seroprevalence curves for the multi-strain structure of influenza A virus
por: Vinh, Dao Nguyen, et al.
Publicado: (2021)

Cannot write session to /tmp/vufind_sessions/sess_dspkt4spp89c25jft0dt0hj8e3