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The Suzuki Reaction Applied to the Synthesis of Novel Pyrrolyl and Thiophenyl Indazoles

The paper describes the Suzuki cross-coupling of a variety of N and C-3 substituted 5-bromoindazoles with N-Boc-2-pyrrole and 2-thiopheneboronic acids. The reactions, performed in the presence of K(2)CO(3), dimethoxyethane and Pd(dppf)Cl(2) as catalyst, gave the corresponding adducts in good yields....

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Detalles Bibliográficos
Autores principales:	Migliorini, Antonella, Oliviero, Chiara, Gasperi, Tecla, Loreto, Maria Antonietta
Formato:	Online Artículo Texto
Lenguaje:	English
Publicado:	MDPI 2012
Materias:	Article
Acceso en línea:	https://www.ncbi.nlm.nih.gov/pmc/articles/PMC6268423/ https://www.ncbi.nlm.nih.gov/pubmed/22508331 http://dx.doi.org/10.3390/molecules17044508

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