Cargando…

4-Thiazolidinones in Heterocyclic Synthesis: Synthesis of Novel Enaminones, Azolopyrimidines and 2-Arylimino-5-arylidene-4-thiazolidinones

The 4-thiazolidinones 3a–d were used as a key intermediates for the synthesis of 2-arylimino-5-arylidene-4-thiazolidinones derivatives 7a–p via nucleophilic addition reactions with the arylidene malononitrile. Moreover the 4-thiazolidinones 3a and 3c condensed with the DMF-DMA to form the correspond...

Descripción completa

Detalles Bibliográficos
Autores principales:	Behbehani, Haider, Ibrahim, Hamada Mohamed
Formato:	Online Artículo Texto
Lenguaje:	English
Publicado:	MDPI 2012
Materias:	Article
Acceso en línea:	https://www.ncbi.nlm.nih.gov/pmc/articles/PMC6268424/ https://www.ncbi.nlm.nih.gov/pubmed/22634845 http://dx.doi.org/10.3390/molecules17066362

Ejemplares similares

The first Q-Tube based high-pressure synthesis of anti-cancer active thiazolo[4,5-c]pyridazines via the [4 + 2] cyclocondensation of 3-oxo-2-arylhydrazonopropanals with 4-thiazolidinones
por: Ibrahim, Hamada Mohamed, et al.
Publicado: (2020)

Author Correction: The first Q-Tube based high-pressure synthesis of anti-cancer active thiazolo[4,5-c]pyridazines via the [4 + 2] cyclocondensation of 3-oxo-2-arylhydrazonopropanals with 4-thiazolidinones
por: Ibrahim, Hamada Mohamed, et al.
Publicado: (2020)

Synthesis of Novel Sulfamethaoxazole 4-Thiazolidinone Hybrids and Their Biological Evaluation
por: Bhat, Mashooq A., et al.
Publicado: (2020)

Synthesis and biological activity evaluation of 5-pyrazoline substituted 4-thiazolidinones
por: Havrylyuk, Dmytro, et al.
Publicado: (2013)

Synthesis and antiviral properties of novel indole-based thiosemicarbazides and 4-thiazolidinones
por: Cihan-Üstündağ, Gökçe, et al.
Publicado: (2016)

Synthesis of Novel Highly Functionalized 4-Thiazolidinone Derivatives from 4-Phenyl-3-thiosemicarbazones
por: Benmohammed, Abdelmadjid, et al.
Publicado: (2014)

Novel 4-Thiazolidinone Derivatives as Anti-Infective Agents: Synthesis, Characterization, and Antimicrobial Evaluation
por: Gupta, Amit, et al.
Publicado: (2016)

Novel 4-thiazolidinone derivatives as agonists of benzodiazepine receptors: Design, synthesis and pharmacological evaluation
por: Faizi, Mehrdad, et al.
Publicado: (2017)

Novel Thiazolidinone-Azole Hybrids: Design, Synthesis and Antimycobacterial Activity Studies
por: Eroglu, Barbaros, et al.
Publicado: (2016)

5-Ene-4-thiazolidinones – An efficient tool in medicinal chemistry
por: Kaminskyy, Danylo, et al.
Publicado: (2017)

Synthesis and Anticancer Activity Evaluation of 5-[2-Chloro-3-(4-nitrophenyl)-2-propenylidene]-4-thiazolidinones
por: Buzun, Kamila, et al.
Publicado: (2021)

Design, Synthesis, Antimicrobial Evaluation and Molecular Modeling Study of 1,2,4-Triazole-Based 4-Thiazolidinones
por: Ahmed, Sahar, et al.
Publicado: (2016)

4-Thiazolidinone Derivatives as MMP Inhibitors in Tissue Damage: Synthesis, Biological Evaluation and Docking Studies
por: Incerti, Matteo, et al.
Publicado: (2018)

Synthesis of Novel Fluorine Compounds Substituted-4-thiazolidinones Derived from Rhodanine Drug as Highly Bioactive Probes
por: Makki, Mohammad S.T., et al.
Publicado: (2019)

4-Thiazolidinone-Bearing Hybrid Molecules in Anticancer Drug Design
por: Roszczenko, Piotr, et al.
Publicado: (2022)

Thiazoles and Thiazolidinones as COX/LOX Inhibitors
por: Liaras, Konstantinos, et al.
Publicado: (2018)

An Efficient and Facile Synthesis of 1,2,4-Aryl Triazoles and 4-Thiazolidinones Bearing 6-Fluorochroman Nucleus
por: Vekariya, Piyush B., et al.
Publicado: (2014)

The design, synthesis, and in vitro trypanocidal and leishmanicidal activities of 1,3-thiazole and 4-thiazolidinone ester derivatives
por: Haroon, Muhammad, et al.
Publicado: (2021)

A Facile Synthesis and Anticancer Activity Evaluation of Spiro[Thiazolidinone-Isatin] Conjugates
por: Kaminskyy, Danylo, et al.
Publicado: (2011)

Synthesis and Characterization of New Thiazolidinones Containing Coumarin Moieties and Their Antibacterial and Antioxidant Activities
por: Hamdi, Naceur, et al.
Publicado: (2012)

An experimental and mechanism study on the regioselective click reaction toward the synthesis of thiazolidinone-triazole
por: Darroudi, Mahdieh, et al.
Publicado: (2021)

Synthesis and biological evaluation of anti-Toxoplasma gondii activity of a novel scaffold of thiazolidinone derivatives
por: Carradori, Simone, et al.
Publicado: (2017)

Antimicrobial and Dyeing Properties of Reactive Dyes with Thiazolidinon-4-one Nucleus
por: Ayalew, Hailemichael, et al.
Publicado: (2014)

In vitro evaluation of new 4-thiazolidinones on invasion and growth of Toxoplasma gondii
por: Molina, Diego A., et al.
Publicado: (2021)

Evaluation of Anticancer and Antibacterial Activity of Four 4-Thiazolidinone-Based Derivatives
por: Skóra, Bartosz, et al.
Publicado: (2022)

On the mechanism of CFTR inhibition by a thiazolidinone derivative
por: Kopeikin, Zoia, et al.
Publicado: (2010)

Antiinflammatory, Analgesic and Antipyretic Activity of Certain Thiazolidinones
por: Taranalli, A. D., et al.
Publicado: (2008)

Development of Thiazolidinones as Fungal Carbonic Anhydrase Inhibitors
por: Güzel-Akdemir, Özlen, et al.
Publicado: (2020)

Design, Synthesis, and Biological Evaluation of Novel Thiazolidinone-Containing Quinoxaline-1,4-di-N-oxides as Antimycobacterial and Antifungal Agents
por: Zhang, Heying, et al.
Publicado: (2020)

The influence of the polymerization approach on the catalytic performance of novel porous poly (ionic liquid)s for green synthesis of pharmaceutical spiro-4-thiazolidinones
por: Elyasi, Zahra, et al.
Publicado: (2020)

Microwave-Assisted Synthesis of some Novel Azoles and Azolopyrimidines as Antimicrobial Agents
por: Gomha, Sobhi M., et al.
Publicado: (2017)

Synthesis and Antimicrobial Evaluation of Some New Thiazoline and Thiazolidinone Derivatives Incorporating [1,2,4]Triazolo[1,5-a]benzimidazole
por: Mahmoud, A. M., et al.
Publicado: (2013)

Design and synthesis of new thiazolidinone/uracil derivatives as antiproliferative agents targeting EGFR and/or BRAF(V600E)
por: Alshammari, Mohammed B., et al.
Publicado: (2022)

Synthesis, Molecular Docking Analysis, and Carbonic Anhydrase Inhibitory Evaluations of Benzenesulfonamide Derivatives Containing Thiazolidinone
por: Zhang, Zuo-Peng, et al.
Publicado: (2019)

Synthesis and Identification of New N,N-Disubstituted Thiourea, and Thiazolidinone Scaffolds Based on Quinolone Moiety as Urease Inhibitor
por: Elshaier, Yaseen A. M. M., et al.
Publicado: (2022)

New 4-Thiazolidinones of Nicotinic Acid with 2-Amino-6-methylbenzothiazole and their Biological Activity
por: Patel, Navin B., et al.
Publicado: (2010)

Structural Optimization and Structure–Activity Relationship of 4-Thiazolidinone Derivatives as Novel Inhibitors of Human Dihydroorotate Dehydrogenase
por: Zeng, Fanxun, et al.
Publicado: (2019)

Mechanochemical Synthesis of Thiazolidinone-Triazoles Derivatives as Antidiabetic Agents: Pharmacokinetics, Molecular Docking, and In Vitro Antidiabetic Properties
por: Taj, M. B., et al.
Publicado: (2023)

Organocatalysis in heterocyclic synthesis: DABCO as a mild and efficient catalytic system for the synthesis of a novel class of quinazoline, thiazolo [3,2-a]quinazoline and thiazolo[2,3-b] quinazoline derivatives
por: Behbehani, Haider, et al.
Publicado: (2013)

Utilisation of Home Laundry Effluent (HLE) as a catalyst for expeditious one-pot aqueous phase synthesis of highly functionalised 4-thiazolidinones
por: Singh, Udaya Pratap, et al.
Publicado: (2013)

Cannot write session to /tmp/vufind_sessions/sess_uugqaurbr51rp7848aave32bee