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(18)F-labeled Pyrazolo[1,5-a]pyrimidine Derivatives: Synthesis from 2,4-Dinitrobenzamide and Tosylate Precursors and Comparative Biological Evaluation for Tumor Imaging with Positron Emission Tomography

We previously reported (18)F-labeled pyrazolo[1,5-a]pyrimidine derivatives: 7-(2-[(18)F]fluoroethylamino)-5-methylpyrazolo[1,5-a]pyrimidine-3-carbonitrile ([(18)F]1) and N-(2-(3-cyano-5-methylpyrazolo[1,5-a]pyrimidin-7-ylamino)ethyl)-2-[(18)F]fluoro-4-nitro- benzamide ([(18)F]2). Preliminary biodist...

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Detalles Bibliográficos
Autores principales:	Xu, Jingli, Liu, Hang, Li, Guixia, He, Yong, Ding, Rui, Wang, Xiao, Feng, Man, Zhang, Shuting, Chen, Yurong, Li, Shilei, Zhao, Mingxia, Li, Yingruo, Qi, Chuanmin, Dang, Yonghong
Formato:	Online Artículo Texto
Lenguaje:	English
Publicado:	MDPI 2012
Materias:	Article
Acceso en línea:	https://www.ncbi.nlm.nih.gov/pmc/articles/PMC6268720/ https://www.ncbi.nlm.nih.gov/pubmed/22453929 http://dx.doi.org/10.3390/molecules17043774

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