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A Convenient One-Pot Preparation of 2-Methyl-3-(phenylthio- methyl)quinolines from Morita-Baylis-Hillman Adducts and Their Oxidation to the Corresponding Sulfones

A convenient one-pot preparation of 2-methyl-3-(phenylthiomethyl)quinolines from Morita-Baylis-Hillman adducts via conjugate addition of thiols followed by reductive cyclization with Fe/AcOH was developed. The 2-methyl-3-(phenylthiomethyl)quinolines were transformed into 2-methyl-3-(phenylsulfonylme...

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Detalles Bibliográficos
Autores principales:	Ramesh, Chintakunta, Lei, Po-Min, Kavala, Veerababurao, Kuo, Chun-Wei, Yao, Ching-Fa
Formato:	Online Artículo Texto
Lenguaje:	English
Publicado:	MDPI 2012
Materias:	Article
Acceso en línea:	https://www.ncbi.nlm.nih.gov/pmc/articles/PMC6268867/ https://www.ncbi.nlm.nih.gov/pubmed/22555297 http://dx.doi.org/10.3390/molecules17055081

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