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A Macrocyclic Peptide that Serves as a Cocrystallization Ligand and Inhibits the Function of a MATE Family Transporter

The random non-standard peptide integrated discovery (RaPID) system has proven to be a powerful approach to discover de novo natural product-like macrocyclic peptides that inhibit protein functions. We have recently reported three macrocyclic peptides that bind to Pyrococcus furiosus multidrug and t...

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Detalles Bibliográficos
Autores principales:	Hipolito, Christopher J., Tanaka, Yoshiki, Katoh, Takayuki, Nureki, Osamu, Suga, Hiroaki
Formato:	Online Artículo Texto
Lenguaje:	English
Publicado:	MDPI 2013
Materias:	Article
Acceso en línea:	https://www.ncbi.nlm.nih.gov/pmc/articles/PMC6270235/ https://www.ncbi.nlm.nih.gov/pubmed/23999725 http://dx.doi.org/10.3390/molecules180910514

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