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TDAE Strategy for the Synthesis of 2,3-Diaryl N-Tosylaziridines

We report herein an original and rapid synthesis of 2,3-diaryl N-tosylaziridines by TDAE strategy starting from ortho- or para-nitro(dichloromethyl)benzene derivatives and N-tosylimines. A mixture of cis/trans isomers was isolated from 1-(dichloromethyl)-4-nitrobenzene, whereas only trans-aziridines...

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Detalles Bibliográficos
Autores principales:	Khoumeri, Omar, Spitz, Cédric, Terme, Thierry, Vanelle, Patrice
Formato:	Online Artículo Texto
Lenguaje:	English
Publicado:	MDPI 2013
Materias:	Communication
Acceso en línea:	https://www.ncbi.nlm.nih.gov/pmc/articles/PMC6270596/ https://www.ncbi.nlm.nih.gov/pubmed/23884113 http://dx.doi.org/10.3390/molecules18077364

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